Compile Data Set for Download or QSAR
maximum 50k data
Found 49 of ec50 data for polymerid = 9460
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430010(CHEMBL2335047)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430008(CHEMBL2335050)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430007(CHEMBL2335051)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430012(CHEMBL357053)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  17nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50381022(CHEMBL2017139)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430011(CHEMBL153043)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430009(CHEMBL2335049)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at LPA1 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148349((3-Octadec-9-enoylamino-propionyl)-phosphonothioic...)
Affinity DataEC50:  40nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430013(CHEMBL364797)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50233165(CHEMBL1222042)
Affinity DataEC50:  80nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as increase in intracellular calcium level measured every 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50170844(CHEMBL187459 | Thiophosphoric acid (E)-octadec-9-e...)
Affinity DataEC50:  193nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50074700(CHEMBL117754 | Phosphoric acid mono-[2-((Z)-octade...)
Affinity DataEC50:  197nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148351(CHEMBL117529 | [3-((Z)-Octadec-9-enoylamino)-propi...)
Affinity DataEC50:  221nMAssay Description:Agonist activity at LPA1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148351(CHEMBL117529 | [3-((Z)-Octadec-9-enoylamino)-propi...)
Affinity DataEC50:  221nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539034(CHEMBL4642952)
Affinity DataEC50:  240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539042(CHEMBL4646737)
Affinity DataEC50:  240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148350(CHEMBL325970 | [3-((Z)-Octadec-9-enoylamino)-thiop...)
Affinity DataEC50:  318nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human LPA1 expressed in LPA1xLPA2 double knockout mouse MEF cells up to 10 uM by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539031(CHEMBL4643262)
Affinity DataEC50:  450nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539036(CHEMBL4636453)
Affinity DataEC50:  500nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50176390((R)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosp...)
Affinity DataEC50:  695nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148352(CHEMBL325288 | [1-Hydroxy-3-((Z)-octadec-9-enoylam...)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 receptor using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539044(CHEMBL4648374)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539046(CHEMBL4636192)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50170848(2-Hexadecanoylamino-3-phosphonooxy-propionic acid ...)
Affinity DataEC50:  1.85E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >1.94E+3nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148355(CHEMBL331661 | [3-((Z)-Octadec-9-enoylamino)-propy...)
Affinity DataEC50:  1.95E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539032(CHEMBL4633208)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539035(CHEMBL4642688)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539030(CHEMBL4647245)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539040(CHEMBL4637403)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539037(CHEMBL4645684)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50176400((R)-2,3-bis(octyloxy)propyl dihydrogen phosphate |...)
Affinity DataEC50:  3.26E+3nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539038(CHEMBL4644847)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539029(CHEMBL4646443)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at recombinant human full-length LPA1 receptor expressed in dhfr- deficient CHO cells assessed as increase in intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539033(CHEMBL4632820)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148353((1-Hydroxy-3-octadec-9-enoylamino-1-phosphono-prop...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148354(CHEMBL117663 | [1-Fluoro-3-((Z)-octadec-9-enoylami...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539043(CHEMBL4648051)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539045(CHEMBL4648653)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50271700(4-(4-(ethoxycarbonyl)styryl)benzenesulfonic acid |...)
Affinity DataEC50: >1.23E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539039(CHEMBL4637898)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50539041(CHEMBL4643694)
Affinity DataEC50:  2.60E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed