Compile Data Set for Download or QSAR
maximum 50k data
Found 160 of ic50 data for polymerid = 1554
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095366(5-(2-Bromo-benzyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095367(5-(2,3-Dimethyl-cyclohexyl)-7-(6-morpholin-4-yl-py...)
Affinity DataIC50:  0.230nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095359(5-[1-(2-Bromo-phenyl)-ethyl]-7-(6-morpholin-4-yl-p...)
Affinity DataIC50:  0.25nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135894(5,6-Bis-(3-fluoro-4-methyl-phenyl)-7-thiophen-2-yl...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135905(5-(4-Bromo-thiophen-2-yl)-6-(3,4-dimethoxy-phenyl)...)
Affinity DataIC50:  0.430nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135900(5,6-Diphenyl-7-thiophen-2-yl-pyrido[2,3-d]pyrimidi...)
Affinity DataIC50:  0.550nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14486((2R,3R,4S,5R)-2-(2-amino-9-iodo-3,5,7-triazabicycl...)
Affinity DataIC50:  0.900nMpH: 7.5 T: 2°CAssay Description:ADK activity was monitored by a radiochemical assay, which measures the conversion of radioactive Ado ([U-14C] adenosine or [2-3H] adenosine) to AMP ...More data for this Ligand-Target Pair
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135888(5-(4-Bromo-thiophen-2-yl)-6-(3,4-dimethoxy-phenyl)...)
Affinity DataIC50:  0.980nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14486((2R,3R,4S,5R)-2-(2-amino-9-iodo-3,5,7-triazabicycl...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14486((2R,3R,4S,5R)-2-(2-amino-9-iodo-3,5,7-triazabicycl...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition of Adenosine kinase of rat brain cytosol.More data for this Ligand-Target Pair
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  1.70nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100580(5-(3-Bromo-phenyl)-7-(6-dimethylamino-pyridin-3-yl...)
Affinity DataIC50:  1.80nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50104168(4-Amino-6-((2R,3R,4S,5R)-5-aminomethyl-3,4-dihydro...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of Adenosine kinase of rat brain cytosol.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117165(5-[(Benzyl-methyl-amino)-methyl]-6-(6-morpholin-4-...)
Affinity DataIC50:  2nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095377(5-Cyclopentyl-7-(6-morpholin-4-yl-pyridin-3-yl)-py...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117169(5-[3-(4-Bromo-phenyl)-propyl]-6-(6-morpholin-4-yl-...)
Affinity DataIC50:  2nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14494(6-{2-[6-(morpholin-4-yl)pyridin-3-yl]ethynyl}-5-(3...)
Affinity DataIC50:  2.5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117175(5-[3-(2-Chloro-phenyl)-propyl]-6-(6-morpholin-4-yl...)
Affinity DataIC50:  2.5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14494(6-{2-[6-(morpholin-4-yl)pyridin-3-yl]ethynyl}-5-(3...)
Affinity DataIC50:  2.5nMpH: 7.5 T: 2°CAssay Description:ADK activity was monitored by a radiochemical assay, which measures the conversion of radioactive Ado ([U-14C] adenosine or [2-3H] adenosine) to AMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090895((2R,3R,4S,5R)-2-[4-(4-Fluoro-phenylamino)-5-phenyl...)
Affinity DataIC50:  2.80nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135891(CHEMBL346622 | [4-Amino-5-(3-bromo-phenyl)-7-thiop...)
Affinity DataIC50:  3nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095379(5-Cyclohexyl-7-(6-morpholin-4-yl-pyridin-3-yl)-pyr...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against intact cell adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095362(5-(2-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135899(5-(3-Bromo-phenyl)-6-(3,4-dimethoxy-phenyl)-7-(4-d...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135898(7-(6-Dimethylamino-pyridin-3-yl)-5,6-diphenyl-pyri...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117164(5-[3-(3-Bromo-phenyl)-propyl]-6-(6-morpholin-4-yl-...)
Affinity DataIC50:  3.5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117154(5-[3-(4-Methoxy-phenyl)-propyl]-6-(6-morpholin-4-y...)
Affinity DataIC50:  3.5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50104164(4-((2R,3R,4S,5R)-5-Aminomethyl-3,4-dihydroxy-tetra...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of Adenosine kinase of rat brain cytosol.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117171(6-(6-Morpholin-4-yl-pyridin-3-ylethynyl)-5-(3-pyri...)
Affinity DataIC50:  4nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135897(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  4nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117155(6-(6-Morpholin-4-yl-pyridin-3-ylethynyl)-5-(3-pyri...)
Affinity DataIC50:  4nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117170(6-(6-Morpholin-4-yl-pyridin-3-ylethynyl)-5-pheneth...)
Affinity DataIC50:  4.5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095384(5-(3-Bromo-phenyl)-7-(4-dimethylamino-phenyl)-pyri...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095373(5-(2,3-Dichloro-phenyl)-7-(6-morpholin-4-yl-pyridi...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135889(5-(3-Bromo-phenyl)-6-(4-fluoro-phenyl)-7-(6-morpho...)
Affinity DataIC50:  5nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135893(5-(3-Chloro-phenyl)-7-(6-dimethylamino-pyridin-3-y...)
Affinity DataIC50:  5nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117173(5-{[(2-Chloro-benzyl)-methyl-amino]-methyl}-6-(6-m...)
Affinity DataIC50:  5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117168(CHEMBL121391 | N*5*-(3-Bromo-benzyl)-N*5*-methyl-6...)
Affinity DataIC50:  5nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095384(5-(3-Bromo-phenyl)-7-(4-dimethylamino-phenyl)-pyri...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095384(5-(3-Bromo-phenyl)-7-(4-dimethylamino-phenyl)-pyri...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against intact cell adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50117162(CHEMBL121415 | N*5*-Methyl-N*5*-(2-methyl-benzyl)-...)
Affinity DataIC50:  6nMAssay Description:Evaluated in vitro for inhibitory activity against Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135904(7-(4-Dimethylamino-phenyl)-5,6-bis-(4-isopropyl-ph...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095358(7-(4-Dimethylamino-phenyl)-5-phenyl-pyrido[2,3-d]p...)
Affinity DataIC50:  7nMAssay Description:Inhibitory activity against intact cell adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095358(7-(4-Dimethylamino-phenyl)-5-phenyl-pyrido[2,3-d]p...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095358(7-(4-Dimethylamino-phenyl)-5-phenyl-pyrido[2,3-d]p...)
Affinity DataIC50:  7nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095372(5-Cyclohexyl-7-(4-dimethylamino-phenyl)-pyrido[2,3...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against intact cell adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095372(5-Cyclohexyl-7-(4-dimethylamino-phenyl)-pyrido[2,3...)
Affinity DataIC50:  8.30nMAssay Description:In vitro inhibition of Adenosine kinase (AK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095364(5-(1-Ethyl-propyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14491(5-(2H-1,3-benzodioxol-5-yl)-6-{2-[4-(dimethylamino...)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:ADK activity was monitored by a radiochemical assay, which measures the conversion of radioactive Ado ([U-14C] adenosine or [2-3H] adenosine) to AMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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