Compile Data Set for Download or QSAR
maximum 50k data
Found 41 of ic50 data for polymerid = 50000292,50000294,50007602,50007794,50007795,50007822
TargetTolloid-like protein 1(Homo sapiens)
Glaxosmithkline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50458762(CHEMBL4207308)
Affinity DataIC50:  100nMAssay Description:Inhibition of PI3Kgamma (2 to 1102) (unknown origin) using diC8-PIP2 as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTolloid-like protein 2(Homo sapiens)
Glaxosmithkline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50458762(CHEMBL4207308)
Affinity DataIC50:  160nMAssay Description:Inhibition of recombinant human N-terminal 6His-tagged TLL2 (26 to 1015 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461717(CHEMBL4225532)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50279578(CHEMBL4177335)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461722(CHEMBL4226440)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461726(CHEMBL4228497)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461718(CHEMBL4227329)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461724(CHEMBL4228556)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461723(CHEMBL4227286)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461715(CHEMBL4227719)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50084726(4-(Biphenyl-4-carbonyl)-1-(4-methoxy-benzenesulfon...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461716(CHEMBL4227787)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461725(CHEMBL4224730)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461730(CHEMBL4225559)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50216823(2-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499820(CHEMBL3740431)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499818(CHEMBL3740110)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461720(CHEMBL4225657)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461733(CHEMBL4229016)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499820(CHEMBL3740431)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461728(CHEMBL4225259)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50216823(2-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461721(CHEMBL4226498)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461731(CHEMBL4225755)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50084737(4-Benzoyl-1-(4-methoxy-benzenesulfonyl)-piperazine...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461729(CHEMBL4225711)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461727(CHEMBL4228238)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461719(CHEMBL4226235)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461732(CHEMBL4228814)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50279577(CHEMBL4166706)
Affinity DataIC50:  7.91E+4nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499818(CHEMBL3740110)
Affinity DataIC50:  7.94E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50063917((2S,3R)-N(4)-[(2S)-3,3-dimethyl-1-(methylamino)-1-...)
Affinity DataIC50:  7.94E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50063917((2S,3R)-N(4)-[(2S)-3,3-dimethyl-1-(methylamino)-1-...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50092158(1,10-phenanthroline | CHEMBL415879 | US10669227, C...)
Affinity DataIC50:  4.70E+5nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499819(CHEMBL3740244)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499819(CHEMBL3740244)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50356193(CHEMBL398206)
Affinity DataIC50:  3.01E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50356189(CHEMBL1910220)
Affinity DataIC50:  3.14E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50241211((E)-1-(3-hydroxy-4-methoxybenzylidene)thiosemicarb...)
Affinity DataIC50:  3.41E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50241210((E)-1-benzylidenethiosemicarbazide | CHEMBL243185 ...)
Affinity DataIC50:  4.22E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas

Curated by ChEMBL
LigandPNGBDBM50356188(CHEMBL391982)
Affinity DataIC50:  4.25E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed