Affinity DataIC50: 100nMAssay Description:Inhibition of PI3Kgamma (2 to 1102) (unknown origin) using diC8-PIP2 as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human N-terminal 6His-tagged TLL2 (26 to 1015 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TA...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow
Curated by ChEMBL
University Of Glasgow
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow
Curated by ChEMBL
University Of Glasgow
Curated by ChEMBL
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow
Curated by ChEMBL
University Of Glasgow
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Plasmodium falciparum 3D7 FLN (55 to 1193 residues) expressed in Escherichia coli BL21 using Dabcyl-HKRHSFRMRG-EDANS as substrate prein...More data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 7.91E+4nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.94E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow
Curated by ChEMBL
University Of Glasgow
Curated by ChEMBL
Affinity DataIC50: 7.94E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 4.70E+5nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow
Curated by ChEMBL
University Of Glasgow
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 3.01E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 3.14E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 3.41E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 4.22E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair
TargetSnake venom metalloproteinase neuwiedase(Bothrops pauloensis)
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Instituto De Ci£Ncias Exatas
Curated by ChEMBL
Affinity DataIC50: 4.25E+6nMAssay Description:Inhibition of Bothrops pauloensis MP1 assessed as reduction in azocaseinolytic activity after 30 minsMore data for this Ligand-Target Pair