Compile Data Set for Download or QSAR
maximum 50k data
Found 51 of ic50 data for polymerid = 50000385,50007327,50007842
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using putrescine as substrate preincubated wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Affinity DataIC50:  59nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Affinity DataIC50:  93nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM43362(MLS000069752 | N,N-dimethylcarbamodithioic acid (d...)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
Affinity DataIC50:  170nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM43362(MLS000069752 | N,N-dimethylcarbamodithioic acid (d...)
Affinity DataIC50:  180nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50232679(CHEMBL4068784 | US11358936, Compound 4-5)
Affinity DataIC50:  214nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged LOXL3 (1 to 753 residues) assessed as reduction in H2O2 production using DAP as substrate pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant human LOXL4 using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM633246((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((5...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 1(Homo sapiens)
Pharmaxis

US Patent
LigandPNGBDBM633246((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((5...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM633249(N-((1-(4-(((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-...)
Affinity DataIC50: <300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM633246((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((5...)
Affinity DataIC50: <300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
Affinity DataIC50:  310nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526727(CHEMBL4568508 | US10807974, Example 100 | US109950...)
Affinity DataIC50:  860nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50266786(CHEMBL4063337)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of recombinant human LOXL3 assessed as reduction of H2O2 production from oxidative deamination of DAP preincubated for 2 hrs followed by s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50:  1.21E+3nMAssay Description:Table 9: The amine oxidase activity was evaluated by measuring Amplex Red fluorescence using commercially available purified, recombinant human LOXL3...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50266787(CHEMBL4092740)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of recombinant human LOXL3 assessed as reduction of H2O2 production from oxidative deamination of DAP preincubated for 2 hrs followed by s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526722(CHEMBL4457897)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526721(CHEMBL4444163 | US10807974, Example 111 | US109950...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463622(CHEMBL4245637)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50266822(CHEMBL4079398)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of recombinant human LOXL3 assessed as reduction of H2O2 production from oxidative deamination of DAP preincubated for 2 hrs followed by s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463622(CHEMBL4245637)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463620(CHEMBL4240937)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 1(Homo sapiens)
Pharmaxis

US Patent
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of recombinant human LOXL1 using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463615(CHEMBL4251179)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526742(CHEMBL4441069)
Affinity DataIC50:  3.85E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526720(CHEMBL4550042)
Affinity DataIC50:  3.86E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463614(CHEMBL4237334)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463617(CHEMBL4238380)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526726(CHEMBL4574361)
Affinity DataIC50:  6.69E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526731(CHEMBL4564074 | US10807974, Example 103 | US109950...)
Affinity DataIC50:  6.78E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526743(CHEMBL4551909)
Affinity DataIC50:  9.31E+3nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50366038(CHEMBL1356238)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463618(CHEMBL4241062)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50501885(CHEMBL4441173 | US10807974, Example 68 | US1099508...)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50366038(CHEMBL1356238)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463613(CHEMBL1927732)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50526728(CHEMBL4463882 | US10807974, Example 155 | US109950...)
Affinity DataIC50:  2.42E+4nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using cadaverine hydrochloride as substrate pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463617(CHEMBL4238380)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463619(CHEMBL4242081)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463621(CHEMBL3144916)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463618(CHEMBL4241062)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463616(CHEMBL4241417)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463614(CHEMBL4237334)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463620(CHEMBL4240937)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463619(CHEMBL4242081)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463621(CHEMBL3144916)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50463615(CHEMBL4251179)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL3 expressed in CHO cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 4(Homo sapiens)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50463613(CHEMBL1927732)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human LOXL4 expressed in baculovirus infected insect cells using diaminopentane as substrate preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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