Compile Data Set for Download or QSAR
maximum 50k data
Found 32 of ic50 data for polymerid = 50000996
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50:  8nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525914(CHEMBL4558285)
Affinity DataIC50:  32nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM113069(US9695194, 5)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human KLK14 using S-2302 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525895(CHEMBL4447752)
Affinity DataIC50:  126nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525904(CHEMBL4461533)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525905(CHEMBL4517343)
Affinity DataIC50:  251nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525912(CHEMBL4543039)
Affinity DataIC50:  316nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525900(CHEMBL4460168)
Affinity DataIC50:  398nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525899(CHEMBL4465265)
Affinity DataIC50:  398nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525917(CHEMBL4579813)
Affinity DataIC50:  794nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM51911((4-isopropoxybenzyl)-[3-(2-methoxyphenyl)-3-(4-met...)
Affinity DataIC50:  970nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM32709((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-met...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525911(CHEMBL4535907)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525903(CHEMBL4436048)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM33453((3-Amino-[1,2,4]triazol-4-yl)-(4-methoxy-phenyl)-m...)
Affinity DataIC50:  3.43E+3nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50522493(CHEMBL4530083)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of recombinant C-terminal 10His-tagged human KLK14 (Gln19 to Met248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525913(CHEMBL4464120)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525918(CHEMBL4473069)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525897(CHEMBL4536142)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM33437((5-amino-3-phenyl-1,2,4-triazol-1-yl)-(3,4-dimetho...)
Affinity DataIC50: >3.00E+4nMpH: 8.0Assay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM33882((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-chl...)
Affinity DataIC50: >3.00E+4nMpH: 8.0Assay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525901(CHEMBL4448315)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525902(CHEMBL4547455)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444599(CHEMBL3099875)
Affinity DataIC50:  8.70E+4nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444600(CHEMBL1462676)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)
Affinity DataIC50:  9.90E+4nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)
Affinity DataIC50:  1.06E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)
Affinity DataIC50:  1.08E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)
Affinity DataIC50:  1.12E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444596(CHEMBL3099883)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed