Compile Data Set for Download or QSAR
maximum 50k data
Found 26 of ic50 data for polymerid = 50002379
LigandPNGBDBM50386308(CHEMBL2047861)
Affinity DataIC50:  118nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386310(CHEMBL2049092)
Affinity DataIC50:  137nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386311(CHEMBL2049093)
Affinity DataIC50:  258nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386292(CHEMBL2047851)
Affinity DataIC50:  263nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386309(CHEMBL2047862)
Affinity DataIC50:  368nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386312(CHEMBL2049094)
Affinity DataIC50:  402nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386294(CHEMBL2049095)
Affinity DataIC50:  488nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386303(CHEMBL2047856)
Affinity DataIC50:  631nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50324539((S)-(-)-9-(4-aminopiperazin-1-yl)-8-fluoro-3-methy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat brain KAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50324539((S)-(-)-9-(4-aminopiperazin-1-yl)-8-fluoro-3-methy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat KAT-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386299(CHEMBL2047852)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386302(CHEMBL2047855)
Affinity DataIC50: >1.33E+3nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386295(CHEMBL2049096)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386298(CHEMBL2049099)
Affinity DataIC50: >4.92E+3nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386307(CHEMBL2047860)
Affinity DataIC50: >6.81E+3nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386296(CHEMBL2049097)
Affinity DataIC50: >7.97E+3nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386306(CHEMBL2047859)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386304(CHEMBL2047857)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386301(CHEMBL2047854)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386300(CHEMBL2047853)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386293(CHEMBL2049100)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386305(CHEMBL2047858)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50386297(CHEMBL2049098)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126149(CHEMBL3629573)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of rat KAT-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126148(CHEMBL3629572)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of rat KAT-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126148(CHEMBL3629572)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of rat liver KAT2 using [3H]-kynurenine incubated for 2 hrs by liquid scintillation spectrometry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed