Compile Data Set for Download or QSAR
maximum 50k data
Found 44 of ic50 data for polymerid = 50005081
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50154254(CHEMBL3775705)
Affinity DataIC50:  112nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50154253(CHEMBL3775377)
Affinity DataIC50:  115nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50154252(CHEMBL3774934)
Affinity DataIC50:  122nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM51911((4-isopropoxybenzyl)-[3-(2-methoxyphenyl)-3-(4-met...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM32709((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-met...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM33453((3-Amino-[1,2,4]triazol-4-yl)-(4-methoxy-phenyl)-m...)
Affinity DataIC50:  990nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM33882((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-chl...)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM33437((5-amino-3-phenyl-1,2,4-triazol-1-yl)-(3,4-dimetho...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50302107(CHEMBL567893 | Grassystatin A)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of kallikrein 5 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human tissue kallikrein-5 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446229(CHEMBL3109060)
Affinity DataIC50:  2.17E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50438170(CHEMBL2407437)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446215(CHEMBL3109169)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446214(CHEMBL3109170)
Affinity DataIC50:  3.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50355088(CHEMBL1834754)
Affinity DataIC50:  5.37E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446216(CHEMBL3109168)
Affinity DataIC50:  5.39E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50355086(CHEMBL1834753)
Affinity DataIC50:  7.29E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataIC50:  9.91E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446227(CHEMBL3109056)
Affinity DataIC50:  9.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataIC50:  9.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)
Affinity DataIC50:  1.17E+5nMAssay Description:Inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)
Affinity DataIC50:  1.17E+5nMAssay Description:Inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)
Affinity DataIC50:  1.27E+5nMAssay Description:Inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)
Affinity DataIC50:  1.31E+5nMAssay Description:Inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446230(CHEMBL3109059)
Affinity DataIC50:  1.57E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446213(CHEMBL3109171)
Affinity DataIC50:  1.57E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446225(CHEMBL3109159)
Affinity DataIC50:  2.23E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446212(CHEMBL3109057)
Affinity DataIC50:  3.21E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataIC50:  3.24E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446223(CHEMBL3109161)
Affinity DataIC50:  3.57E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50355087(CHEMBL1833982)
Affinity DataIC50:  3.67E+5nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446222(CHEMBL3109162)
Affinity DataIC50:  3.77E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446217(CHEMBL3109167)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50446226(CHEMBL3109158)
Affinity DataIC50:  5.21E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed