Compile Data Set for Download or QSAR
maximum 50k data
Found 249 of kd data for polymerid = 1325
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50460772(CHEMBL4225923)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to Aurora A (unknown origin) after 45 mins by fluorescence-based thermal stability shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50460773(CHEMBL4227082)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to Aurora A (unknown origin) after 45 mins by fluorescence-based thermal stability shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM109208(2-[(1E,3E)-5-[(2E)-3-(3-{[(5R)-5-carbamoyl-5-{[4- ...)
Affinity DataKd:  0.200nMT: 2°CAssay Description:A stock solution was prepared containing complex of Aurora A and Compound I (final total concentrations of 6nM and 5nM, respectively). Separately, se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM109206(2-[(1E,3E)-5-[(2E)-3-(3-{[(5R)-5-carbamoyl-5-[(4- ...)
Affinity DataKd:  0.273nMT: 2°CAssay Description:A stock solution was prepared containing complex of Aurora A and Compound I (final total concentrations of 6nM and 5nM, respectively). Separately, se...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106623(CHEMBL3600871)
Affinity DataKd:  0.440nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKd:  0.501nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106624(CHEMBL3600870)
Affinity DataKd:  0.730nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to AURKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106631(CHEMBL3600653)
Affinity DataKd:  1.90nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106630(CHEMBL3600760)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394776(CHEMBL2163388)
Affinity DataKd:  2.5nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106625(CHEMBL3600869)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394789(CHEMBL2163400)
Affinity DataKd:  2.80nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKd:  3.90nMAssay Description:Binding constant for AURKA kinase domainMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394783(CHEMBL2163390)
Affinity DataKd:  4nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394788(CHEMBL2163401)
Affinity DataKd:  4nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394782(CHEMBL2163391)
Affinity DataKd:  4nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKd:  4nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKd:  4.10nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKd:  4.10nMAssay Description:Binding constant for AURKA kinase domainMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394778(CHEMBL2163395)
Affinity DataKd:  4.20nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394799(CHEMBL2163407)
Affinity DataKd:  4.5nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352328(CHEMBL1822648)
Affinity DataKd:  5nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50198027(CHEMBL3921246)
Affinity DataKd:  5nMAssay Description:Binding affinity to human Aurora A kinase expressed in Escherichia coli BL21 cells incubated for 1 hr by active site directed binding competition ass...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352325(CHEMBL1822651)
Affinity DataKd:  5nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394795(CHEMBL2163411)
Affinity DataKd:  5.10nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM109207(Compound II: Ac-D-Arg6-D-Lys(PromoFluor 647)-D-Lys...)
Affinity DataKd:  5.20nMT: 2°CAssay Description:A stock solution was prepared containing complex of Aurora A and Compound I (final total concentrations of 6nM and 5nM, respectively). Separately, se...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394777(CHEMBL2163387)
Affinity DataKd:  5.60nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106627(CHEMBL3600764)
Affinity DataKd:  5.70nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394785(CHEMBL2163404)
Affinity DataKd:  5.80nMAssay Description:Binding affinity to Aurora kinase A catalytic domain by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352327(CHEMBL1822649)
Affinity DataKd:  6nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106626(CHEMBL3600868)
Affinity DataKd:  6.10nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394781(CHEMBL2163392)
Affinity DataKd:  6.30nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394786(CHEMBL2163403)
Affinity DataKd:  6.30nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394784(CHEMBL2163389)
Affinity DataKd:  6.40nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)
Affinity DataKd:  6.5nMAssay Description:Binding constant for AURKA kinase domainMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)
Affinity DataKd:  6.5nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50106628(CHEMBL3600763)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to purified recombinant full-length Aurora A (unknown origin) by fluorescence polarisation/anisotropy based equilibrium binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)
Affinity DataKd:  6.5nMAssay Description:Binding constant for AURKA kinase domainMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352298(CHEMBL1822661)
Affinity DataKd:  7nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352300(CHEMBL1822487)
Affinity DataKd:  7nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352303(CHEMBL1822490)
Affinity DataKd:  7nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352323(CHEMBL1822653)
Affinity DataKd:  7nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50401421(CHEMBL2207503)
Affinity DataKd:  7.5nMAssay Description:Binding affinity to Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM247371(US9447092, 1)
Affinity DataKd:  7.5nMAssay Description:The kinase selectivity was assessed by profiling Example 1 in a 442-kinase panel (386 non-mutant kinases) at a concentration of 1 μM using the K...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352324(CHEMBL1822652)
Affinity DataKd:  8nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352326(CHEMBL1822650)
Affinity DataKd:  8nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352307(CHEMBL1822640)
Affinity DataKd:  8nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50352309(CHEMBL1822638)
Affinity DataKd:  8nMAssay Description:Binding affinity to Aurora A kinase catalytic domain by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50394786(CHEMBL2163403)
Affinity DataKd:  8.80nMAssay Description:Binding affinity to Aurora kinase A catalytic domain by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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