Affinity DataKd: 0.0302nMAssay Description:Binding affinity to human recombinant NK1 receptor expressed in CHO cells assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 0.180nMAssay Description:Scatchard analysis at concentration of the 3 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 0.970nMAssay Description:Scatchard analysis at concentration of the 1 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Scatchard analysis at concentration of the 10 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 3.98nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 5.37nMAssay Description:Competitive inhibition of wild type human NK1 receptor expressed in HEK293 cells assessed as decrease in SP1-induced [3H]IP accumulation after 20 min...More data for this Ligand-Target Pair
Affinity DataKd: 15.8nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 31.6nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 540nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 631nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 670nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 860nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 3.80E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair