Affinity DataKd: 0.0302nMAssay Description:Binding affinity to human recombinant NK1 receptor expressed in CHO cells assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 0.180nMAssay Description:Scatchard analysis at concentration of the 3 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 0.320nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 0.970nMAssay Description:Scatchard analysis at concentration of the 1 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Scatchard analysis at concentration of the 10 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 3.98nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 5.37nMAssay Description:Competitive inhibition of wild type human NK1 receptor expressed in HEK293 cells assessed as decrease in SP1-induced [3H]IP accumulation after 20 min...More data for this Ligand-Target Pair
Affinity DataKd: 15.8nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 31.6nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 39.8nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisinMore data for this Ligand-Target Pair
Affinity DataKd: 126nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against Tachykinin receptor 1 in guinea pig myenteric plexus longitudinal muscle st...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
Affinity DataKd: 251nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisinMore data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 398nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
Affinity DataKd: 501nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
Affinity DataKd: 540nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 631nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 670nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 860nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.26E+3nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisin (mean +/-, n=4)More data for this Ligand-Target Pair
Affinity DataKd: 3.80E+3nMAssay Description:Binding affinity towards Tachykinin receptor 1, activity expressed as KdMore data for this Ligand-Target Pair