Compile Data Set for Download or QSAR
maximum 50k data
Found 55 of kd data for polymerid = 49000773,7531
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)
Affinity DataKd:  11nMAssay Description:TP_TRANSPORTER: binding in plasma membranes from CEM/VLB1.0 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423806(CHEMBL1822225)
Affinity DataKd:  15nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423808(CHEMBL1822227)
Affinity DataKd:  25nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423817(CHEMBL165950)
Affinity DataKd:  33nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423801(CHEMBL164699)
Affinity DataKd:  36nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423807(CHEMBL1822226)
Affinity DataKd:  45nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50095341(3,5,7-Trihydroxy-2-(4-octyl-phenyl)-chromen-4-one ...)
Affinity DataKd:  58nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423802(CHEMBL165418)
Affinity DataKd:  68nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50420186(ZOSUQUIDAR | ZOSUQUIDAR TRIHYDROCHLORIDE)
Affinity DataKd:  73nMAssay Description:TP_TRANSPORTER: binding in membrane vesicle from CEM/VLB100 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423815(CHEMBL1822217)
Affinity DataKd:  151nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423816(CHEMBL193777)
Affinity DataKd:  200nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423804(CHEMBL191602)
Affinity DataKd:  200nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423797(CHEMBL164060)
Affinity DataKd:  209nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423811(CHEMBL1822218)
Affinity DataKd:  209nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423812(CHEMBL1822219)
Affinity DataKd:  219nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423798(CHEMBL166131)
Affinity DataKd:  282nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423805(CHEMBL1822224)
Affinity DataKd:  282nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423803(CHEMBL1822223)
Affinity DataKd:  302nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423799(CHEMBL165452)
Affinity DataKd:  339nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423810(CHEMBL189433)
Affinity DataKd:  447nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423809(CHEMBL1822228)
Affinity DataKd:  708nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423800(CHEMBL165621)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423796(CHEMBL165408)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50095339(3,5,7-Trihydroxy-2-(4-iodo-phenyl)-chromen-4-one |...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50338977(5-Hydroxy-6-methyl-7-methoxy-flavone | 5-Hydroxy-7...)
Affinity DataKd:  1.29E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423813(CHEMBL1822220)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423795(CHEMBL1822222)
Affinity DataKd:  2.19E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataKd:  3.00E+3nMAssay Description:TP_TRANSPORTER: binding in membrane vesicle from CEM/VLB100 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423792(CHEMBL163960)
Affinity DataKd:  3.09E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50095342(2-(2,4-Dichloro-phenyl)-3,5,7-trihydroxy-chromen-4...)
Affinity DataKd:  3.98E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50084978(3,5,7-trihydroxy-2-(4-methoxyphenyl)-4H-chromen-4-...)
Affinity DataKd:  4.47E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50049391(3,5,7-Trihydroxyflavone | 3,5,7-triOH-flavone | 3,...)
Affinity DataKd:  5.89E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423794(CHEMBL1821732)
Affinity DataKd:  6.31E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423793(NSC-80687 | TECHTOCHRYSIN)
Affinity DataKd:  6.31E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataKd:  6.76E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50095340(2-(4-Fluoro-phenyl)-3,5,7-trihydroxy-chromen-4-one...)
Affinity DataKd:  6.76E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKd:  7.08E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50423814(CHEMBL1822221)
Affinity DataKd:  8.91E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM7461(5,7-dihydroxy-2-phenyl-4H-chromen-4-one | 5,7-dihy...)
Affinity DataKd:  8.91E+3nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50187668(3-Hydroxyflavone | 3-Hydroxyflavone (12) | 3-hydro...)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to ABCB1 nucleotide binding domain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514163(CHEMBL4568985)
Affinity DataKd:  2.01E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514155(CHEMBL4553676)
Affinity DataKd:  2.16E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514161(CHEMBL4469705)
Affinity DataKd:  2.22E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514162(CHEMBL4446420)
Affinity DataKd:  2.28E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514157(CHEMBL4552725)
Affinity DataKd:  2.29E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514159(CHEMBL4476464)
Affinity DataKd:  2.31E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514164(CHEMBL4437065)
Affinity DataKd:  2.41E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514158(CHEMBL4526913)
Affinity DataKd:  2.56E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Institute Of Parasitology Of Mcgill University

Curated by ChEMBL
LigandPNGBDBM50514165(CHEMBL4438522)
Affinity DataKd:  2.57E+4nMAssay Description:Inhibition of spin-labelled adenine nucleotide interaction with human P-gp expressed in Escherichia coli BL21 (DE3) assessed as apparent dissociation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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