Affinity DataKd: 0.600nMAssay Description:Binding affinity to mGluR5 ligand binding site 1 in Sprague-Dawley rat brain P2 membrane after 45 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKd: 2.25nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 2.30nMAssay Description:Binding affinity at mGluR5 in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counter in absence of MPEPMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counter in presence of 10 nM MPEPMore data for this Ligand-Target Pair
Affinity DataKd: 7.20nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counter in presence of 20 nM MPEPMore data for this Ligand-Target Pair
Affinity DataKd: 8.60nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 9.40nMAssay Description:Binding affinity to mGluR5 in Sprague-Dawley rat striatum after 60 mins by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataKd: 13.7nMAssay Description:Binding affinity to mGluR5 ligand binding site 2 in Sprague-Dawley rat brain P2 membrane after 45 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKd: 70nMAssay Description:Binding affinity to mGluR5 receptor in Sprague-Dawley rat brain by beta countingMore data for this Ligand-Target Pair