Compile Data Set for Download or QSAR
maximum 50k data
Found 73 of ki data for polymerid = 49000396,49000413
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50170601((1R,10S)-9-oxa-4,13-diazatetracyclo[11.2.1.0^{1,10...)
Affinity DataKi:  116nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  151nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
Targacept

Curated by PDSP Ki Database
LigandPNGBDBM86311(CAS_485-35-8 | Cytisine | Cytisine-(-) | NSC_22407...)
Affinity DataKi:  176nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  187nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  220nMAssay Description:In vitro Binding affinity towards alpha-3 (PC12) nAChR was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
Affinity DataKi:  730nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50254482(3-(dimethylamino)butyl benzyl(methyl)carbamate | C...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50061565((+)Methyl-(2,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl...)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50170601((1R,10S)-9-oxa-4,13-diazatetracyclo[11.2.1.0^{1,10...)
Affinity DataKi:  1.79E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50254486(3-(dimethylamino)butyl 2-hydroxyethylcarbamate | C...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50096712(3-(1H-Indole-3-carbonyloxy)-8,8-dimethyl-8-azonia-...)
Affinity DataKi:  2.30E+3nMAssay Description:In vitro Binding affinity towards alpha-3 (PC12) nAChR was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50254483(3-(dimethylamino)butyl carbamate | CHEMBL449334)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50254542(CHEMBL468903 | O-3-(dimethylamino)butyl dimethylca...)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50254485(3-(dimethylamino)butyl propylcarbamate | CHEMBL466...)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50254541(5-(dimethylamino)-N,N-dimethylhex-2-enamide | CHEM...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50107863((-)-cytisine | (1R,9R)-7,11-diazatricyclo[7.3.1.0~...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50061562((12R,13aR)-12-Methoxy-1,4,5,6,9,11,12,13-octahydro...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50061567(1,1-Dimethyl-4-phenyl-piperazin-1-ium | CHEMBL1347...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM85207(CAS_123990 | NSC_123990 | Suberyldicholine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50159165((2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50159165((2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86199(CAS_595 | CAS_67678 | D-cystine | L-cystine | NSC_...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86196(D-homocysteic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86197(D-homocysteine sulfinic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86205(D-homocysteine thiolactone)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86195(CAS_6137 | CAS_84815 | D-methionine | L-methionine...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86202(CAS_778 | DL-homocysteine | NSC_778)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM85473(L-Cysteic acid, 8 | L-cysteic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86203(CAS_5862 | L-cysteine | NSC_5862)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86194(CAS_109 | L-cysteine sulfinic acid | NSC_109)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86199(CAS_595 | CAS_67678 | D-cystine | L-cystine | NSC_...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50220147((S)-2-amino-4-sulfobutanoic acid | CHEMBL230951 | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86201(L-homocysteine sulfinic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86198(CAS_134505 | L-homocysteine thiolactone | NSC_1345...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86195(CAS_6137 | CAS_84815 | D-methionine | L-methionine...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86199(CAS_595 | CAS_67678 | D-cystine | L-cystine | NSC_...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86196(D-homocysteic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86197(D-homocysteine sulfinic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86205(D-homocysteine thiolactone)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86195(CAS_6137 | CAS_84815 | D-methionine | L-methionine...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86202(CAS_778 | DL-homocysteine | NSC_778)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM85473(L-Cysteic acid, 8 | L-cysteic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86203(CAS_5862 | L-cysteine | NSC_5862)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86194(CAS_109 | L-cysteine sulfinic acid | NSC_109)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86199(CAS_595 | CAS_67678 | D-cystine | L-cystine | NSC_...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50220147((S)-2-amino-4-sulfobutanoic acid | CHEMBL230951 | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM86201(L-homocysteine sulfinic acid)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 73 total ) | Next | Last >>
Jump to: