Compile Data Set for Download or QSAR
maximum 50k data
Found 131 of ki data for polymerid = 49000716,50006057
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120625(CHEMBL3618330)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50241083(6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1...)
Affinity DataKi:  0.340nMAssay Description:Antagonist activity at rat MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120624(CHEMBL3618324)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120635(CHEMBL3618325)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219036(CHEMBL388440 | N-{3-[1-(3-{[hydroxy(diphenyl)acety...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219040(CHEMBL429464 | N-{3-[1-(3-{[bis(4-fluorophenyl)ace...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50094880(CHEMBL3589145)
Affinity DataKi:  0.800nMAssay Description:Antagonist activity at rat MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189584((R)-6-(4-chlorophenyl)-2-(6-(3-(dimethylamino)pyrr...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189587((S)-6-(4-chlorophenyl)-2-(6-(3-(dimethylamino)pyrr...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189581((S)-6-(4-chlorophenyl)-2-(6-(3-(methylamino)pyrrol...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189592((R)-2-(4-methoxyphenyl)-6-(6-(3-(methylamino)pyrro...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120628(CHEMBL3618334)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219026(CHEMBL243338 | N-{3-[1-(3-{[bis(4-fluorophenyl)ace...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120796(CHEMBL3618363)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120676(CHEMBL3618340)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189589((R)-6-(4-chlorophenyl)-2-(6-(3-(methylamino)pyrrol...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189582((S)-6-(4-chlorophenyl)-2-(6-(3-(pyrrolidin-1-ylami...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120629(CHEMBL3618336)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219035(CHEMBL243355 | N-{5-[1-(3-{[bis(4-fluorophenyl)ace...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219047(CHEMBL245231 | N-(3-(1-(4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189578((R)-2-(4-chlorophenyl)-6-(6-(3-(methylamino)pyrrol...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219023(CHEMBL243138 | N-{3-[1-(3-diphenylacetylamino-prop...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189579((S)-6-(4-chlorophenyl)-2-(6-(3-(ethylamino)pyrroli...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219029(CHEMBL390679 | N-{3-[1-(2-diphenylacetylamino-ethy...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219037(1-(4-fluorophenyl)-N-(3-{4-[5-(isobutyrylamino)-2-...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189593((S)-2-(4-fluorophenyl)-6-(6-(3-(methylamino)pyrrol...)
Affinity DataKi:  2nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  2nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219053(CHEMBL242004 | N-(3-{1-4-(3,4-difluorophenoxy)benz...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120670(CHEMBL3618338)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219044(CHEMBL243128 | N-{3-[1-(3-{[bis(4-chlorophenyl)ace...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353455(CHEMBL1830049)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353456(CHEMBL1830050)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189594((R)-2-(4-fluorophenyl)-6-(6-(3-(methylamino)pyrrol...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120634(CHEMBL3618326)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189591((R)-2-(4-ethylphenyl)-6-(6-(3-(methylamino)pyrroli...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120633(CHEMBL3618327)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219025(CHEMBL243578 | N-{3-[1-(3-{[bis(4-fluorophenyl)ace...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219042(CHEMBL242689 | N-[3-(1-{3-[(diphenylacetyl)amino]p...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189586((S)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189576((R)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50094885(CHEMBL3588863)
Affinity DataKi:  3.80nMAssay Description:Antagonist activity at rat MCHR1 assessed as 2-(4-chlorophenyl)-5-(4-(2-hydroxy-2-methylpropoxy)-3-methoxyphenyl)-4,5-dihydropyrrolo[3,4-c]pyrazol-6(...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219031(1-(4-fluorophenyl)-N-(3-{4-[5-(isobutylamino)-2-me...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120675(CHEMBL3618339)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50107746(CHEMBL3600828)
Affinity DataKi:  4nMAssay Description:Antagonist activity against rat MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353453(CHEMBL1830047)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189583((S)-6-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50120674(CHEMBL3618337)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125I][Phe13,Tyr19]-MCH from rat MCHR1 by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353457(CHEMBL1830051)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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