Compile Data Set for Download or QSAR
maximum 50k data
Found 63 of ki data for polymerid = 50000019,50000462
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50049260(3-Hydrazinomethyl-phenol | CHEMBL352205)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50049259(CHEMBL160520 | Methyl-hydrazine)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibitory activity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50024970((2E)-4-ammonio-2-(hydroxymethyl)but-2-enoate | CHE...)
Affinity DataKi:  5.00E+3nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50561618(CHEMBL4746439)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085233(3-Amino-4-fluoro-cyclopentanecarboxylic acid | CHE...)
Affinity DataKi:  1.20E+4nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50024968((2Z)-4-ammonio-2-(fluoromethyl)but-2-enoate | CHEM...)
Affinity DataKi:  1.90E+4nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50024969((2Z)-4-ammonio-2-(chloromethyl)but-2-enoate | CHEM...)
Affinity DataKi:  2.40E+4nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50561615(CHEMBL4747359)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50135932((1S,3S)-3-Amino-4-difluoromethylene-cyclopentaneca...)
Affinity DataKi:  3.10E+4nMAssay Description:Tested for inhibitory activity of the compound against gamma-aminobutyric acid aminotransferase from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082743((1R,4S)-4-Amino-cyclopent-2-enecarboxylic acid | C...)
Affinity DataKi:  4.00E+4nMAssay Description:Reversible inhibition of pig brain GABA-AT using GABA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082743((1R,4S)-4-Amino-cyclopent-2-enecarboxylic acid | C...)
Affinity DataKi:  5.20E+4nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085233(3-Amino-4-fluoro-cyclopentanecarboxylic acid | CHE...)
Affinity DataKi:  5.30E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50135932((1S,3S)-3-Amino-4-difluoromethylene-cyclopentaneca...)
Affinity DataKi:  5.90E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085239(4-Amino-3,3-difluoro-cyclopentanecarboxylic acid |...)
Affinity DataKi:  1.90E+5nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50118886(4-Amino-hex-5-enoic acid | CHEMBL89598 | US1018980...)
Affinity DataKi:  2.90E+5nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50015034(3-Carboxy-1-fluoromethyl-propyl-ammonium | 4-Amino...)
Affinity DataKi:  3.95E+5nMpH: 8.5Assay Description:Compound was tested for inhibitory constant of Gamma-amino-N-butyrate transaminase in pig brain at pH of 8.5 and 25 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50015034(3-Carboxy-1-fluoromethyl-propyl-ammonium | 4-Amino...)
Affinity DataKi:  4.00E+5nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085233(3-Amino-4-fluoro-cyclopentanecarboxylic acid | CHE...)
Affinity DataKi:  4.30E+5nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082744(4-Amino-cyclopent-2-enecarboxylic acid | CHEMBL358...)
Affinity DataKi:  6.00E+5nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50015035(3-Carboxy-1-fluoromethyl-2-phenyl-propyl-ammonium;...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminase in pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082745((R)-4-Amino-cyclopent-1-enecarboxylic acid | CHEMB...)
Affinity DataKi:  1.20E+6nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50199994((1R,4S)-4-amino-3-fluoro-cyclopent-2-ene carboxyli...)
Affinity DataKi:  1.30E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391518(CHEMBL2147351)
Affinity DataKi:  1.35E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391514(CHEMBL2147347)
Affinity DataKi:  1.40E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391519(CHEMBL2147352)
Affinity DataKi:  1.59E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085236(3-Amino-4-bromo-2-fluoro-cyclopentanecarboxylic ac...)
Affinity DataKi:  1.60E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391517(CHEMBL2147350)
Affinity DataKi:  1.64E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50025199(3-Carboxy-1-fluoromethyl-allyl-ammonium)
Affinity DataKi:  2.00E+6nMpH: 6.5Assay Description:Compound was tested for inhibitory constant of Gamma-amino-N-butyrate transaminase in pig brain at pH of 6.5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391516(CHEMBL2147349)
Affinity DataKi:  2.14E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391520(CHEMBL2147353)
Affinity DataKi:  2.27E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM17663((2S)-2-amino-3-(sulfooxy)propanoic acid | L-SOS | ...)
Affinity DataKi:  2.40E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391515(CHEMBL2147348)
Affinity DataKi:  2.49E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082746((1S,4R)-4-Amino-cyclopent-2-enecarboxylic acid | C...)
Affinity DataKi:  2.70E+6nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50199991((1R,4S)-4-amino-3-pentafluoroethyl-cyclopent-2-ene...)
Affinity DataKi:  2.80E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50391521(CHEMBL2147354)
Affinity DataKi:  2.86E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085236(3-Amino-4-bromo-2-fluoro-cyclopentanecarboxylic ac...)
Affinity DataKi:  3.14E+6nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50118886(4-Amino-hex-5-enoic acid | CHEMBL89598 | US1018980...)
Affinity DataKi:  3.20E+6nMAssay Description:Tested for inhibitory activity of the compound against gamma-aminobutyric acid aminotransferase from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085234(3-Amino-4-bromo-cyclopentanecarboxylic acid | CHEM...)
Affinity DataKi:  3.60E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50199992((1R,4S)-4-amino-3-trifluoromethyl-cyclopent-2-ene ...)
Affinity DataKi:  4.11E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50199989((1S,3S)-3-amino-4-(2,2,2-trifluoro-1-trifluorometh...)
Affinity DataKi:  4.20E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085241(3-Amino-2,4-dibromo-cyclopentanecarboxylic acid | ...)
Affinity DataKi:  4.20E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085235(3-Amino-2-bromo-4-fluoro-cyclopentanecarboxylic ac...)
Affinity DataKi:  4.70E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50280206((2S)-2-amino-2-methyl-3-(phosphonooxy)propanoic ac...)
Affinity DataKi:  5.70E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50085238(3-Amino-4-bromo-2-hydroxy-cyclopentanecarboxylic a...)
Affinity DataKi:  5.90E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50561616(CHEMBL4758952)
Affinity DataKi:  6.01E+6nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082127(3-(ammoniomethyl)-2,6-difluorobenzenolate | 3-Amin...)
Affinity DataKi:  6.30E+6nMAssay Description:Competitive inhibition of pig brain GABA aminotransferase by Dixon/Cornish-Bowden plot analysis in presence of GABAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50082127(3-(ammoniomethyl)-2,6-difluorobenzenolate | 3-Amin...)
Affinity DataKi:  6.30E+6nMAssay Description:The compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50280205((R)-2-Amino-3-chloro-2-methyl-propionic acid | CHE...)
Affinity DataKi:  6.50E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50280203((R)-2-Amino-3-fluoro-2-methyl-propionic acid | CHE...)
Affinity DataKi:  6.80E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50199993((1S,3S)-(Z)-3-amino-4-(2,2,2-trifluoroethylidene)c...)
Affinity DataKi:  7.74E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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