Compile Data Set for Download or QSAR
maximum 50k data
Found 25 of ki data for polymerid = 50000044,50000046,50007558,50007713,50007926,50007968,50007969,50007970
TargetBeta-lactamase 1(Bacillus cereus)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50450973(CHEMBL4209255)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of Bacillus cereus beta-lactamase AmpC using CENTA as substrate up to 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase 1(Bacillus cereus)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50450974(CHEMBL4206040)
Affinity DataKi:  0.200nMAssay Description:Inhibition of Bacillus cereus beta-lactamase AmpC using CENTA as substrate up to 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase 1(Bacillus cereus)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50450969(CHEMBL4217629)
Affinity DataKi:  0.800nMAssay Description:Inhibition of Bacillus cereus beta-lactamase AmpC using CENTA as substrate up to 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase 1(Bacillus cereus)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50450975(CHEMBL4204887)
Affinity DataKi:  1.30nMAssay Description:Inhibition of Bacillus cereus beta-lactamase AmpC using CENTA as substrate up to 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA by competitive inhibition assayMore data for this Ligand-Target Pair
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50486725(CHEMBL2236666)
Affinity DataKi:  1.19E+4nMAssay Description:Inhibition of Citrobacter freundii beta-lactamase SHV-95More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 7.0More data for this Ligand-Target Pair
TargetBeta-lactamase(Acinetobacter baumannii)TBA
LigandPNGBDBM50486725(CHEMBL2236666)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase SHV-48More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50486723(PENEM-2)
Affinity DataKi:  2.96E+4nMAssay Description:Inhibition of Citrobacter freundii beta-lactamase SHV-95More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Acinetobacter baumannii)TBA
LigandPNGBDBM50486723(PENEM-2)
Affinity DataKi:  3.47E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase SHV-48More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 8.0More data for this Ligand-Target Pair
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  4.60E+4nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 7.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50486724(PENEM-1)
Affinity DataKi:  4.62E+4nMAssay Description:Inhibition of Citrobacter freundii beta-lactamase SHV-95More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Acinetobacter baumannii)TBA
LigandPNGBDBM50486724(PENEM-1)
Affinity DataKi:  5.44E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase SHV-48More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 8.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  1.08E+5nMAssay Description:Inhibition of Citrobacter freundii beta-lactamase SHV-95More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 9.0More data for this Ligand-Target Pair
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26115(CHEMBL286204 | Quinolinate | Quinolinic acid | pyr...)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Acinetobacter baumannii)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  2.27E+5nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase SHV-48More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26114(CHEMBL88972 | pyridine carboxylate, 6b | pyridine-...)
Affinity DataKi:  4.20E+5nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  4.40E+5nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 10.0More data for this Ligand-Target Pair
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM26117(pyridine carboxylate, 6e | pyridine-3,4-dicarboxyl...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 10.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed