Affinity DataKi: 0.0417nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.0537nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.0661nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.324nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.977nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]RX 821002 from human recombinant adrenergic alpha-2A receptor expressed in CHO cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to alpha2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to alpha2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [3H]-rauwolscine from recombinant human alpha2A adrenergic receptor stably expressed in MDCK cell membranes measured after 90 mins by...More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to human adrenergic alpha 2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Activity of compound against Alpha-2A (ADRA2A) adrenergic receptor by displacement of [3H]-rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 193nMAssay Description:Binding affinity to alpha2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 221nMAssay Description:Displacement of [3H]-rauwolscine from recombinant human alpha2A adrenergic receptor stably expressed in MDCK cells measured after 90 mins by microbet...More data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Displacement of [3H]-Rauwolscine from human recombinant adrenergic Alpha2A receptor expressed in stable MDCK cells after 90 mins by microbeta scintil...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [3H] RX821002 from alpha2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 531nMAssay Description:Binding affinity to alpha 2A adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 537nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 537nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Displacement of [3H]RX 821002 from recombinant human alpha2A receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 603nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 708nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 860nMAssay Description:Displacement of [3H] RX821002 from alpha2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity to adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Activity of compound against Alpha-2A (ADRA2A) adrenergic receptor by displacement of [3H]-rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+3nMAssay Description:Binding affinity to human alpha2A receptor expressed in MDCK cells by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+3nMAssay Description:Binding affinity to human alpha2A receptor expressed in MDCK cells by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]RX821002 from alpha-2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.24E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [3H]RX821002 from alpha-2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of [3H]RX 821002 from recombinant human alpha2A receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [3H]-rauwolscine from recombinant human alpha2A adrenergic receptor stably expressed in MDCK cells measured after 90 mins by microbet...More data for this Ligand-Target Pair
Affinity DataKi: 3.36E+3nMAssay Description:Displacement of [3H] NECA from human adrenergic alpha 2A receptor expressed in MDCK cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [3H]-rauwolscine from recombinant human alpha2A adrenergic receptor stably expressed in MDCK cells measured after 90 mins by microbet...More data for this Ligand-Target Pair
Affinity DataKi: 3.72E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 3.97E+3nMAssay Description:Binding affinity to alpha2a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.37E+3nMAssay Description:Activity of compound against Alpha-2A (ADRA2A) adrenergic receptor by displacement of [3H]-rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 4.57E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair