TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 541nMAssay Description:Binding affinity to biotinylated AAK1 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 5.30E+4nMAssay Description:Binding affinity to C-terminal AVI-tagged AAK1 (unknown origin) (31 to 396 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 7.80E+4nMAssay Description:Binding affinity to C-terminal AVI-tagged AAK1 (unknown origin) (31 to 396 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to C-terminal AVI-tagged AAK1 (unknown origin) (31 to 396 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair