Compile Data Set for Download or QSAR
maximum 50k data
Found 833 of ki data for polymerid = 554
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50035105(1'-{4-[1-(4-fluorophenyl)-1H-3-indolyl]butyl}spiro...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50216056((N-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349368(US10207991, Ex. Cpd. No. 11 | US10611728, Example ...)
Affinity DataKi:  0.440nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349368(US10207991, Ex. Cpd. No. 11 | US10611728, Example ...)
Affinity DataKi:  0.440nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349368(US10207991, Ex. Cpd. No. 11 | US10611728, Example ...)
Affinity DataKi:  0.440nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349368(US10207991, Ex. Cpd. No. 11 | US10611728, Example ...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349518(US10207991, Ex. Cpd. No. 34 | US10611728, Example ...)
Affinity DataKi:  0.530nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349518(US10207991, Ex. Cpd. No. 34 | US10611728, Example ...)
Affinity DataKi:  0.530nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349518(US10207991, Ex. Cpd. No. 34 | US10611728, Example ...)
Affinity DataKi:  0.530nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50540826(CHEMBL4647871)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349505(US10207991, Ex. Cpd. No. 20 | US10611728, Example ...)
Affinity DataKi:  0.670nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349505(US10207991, Ex. Cpd. No. 20 | US10611728, Example ...)
Affinity DataKi:  0.670nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349505(US10207991, Ex. Cpd. No. 20 | US10611728, Example ...)
Affinity DataKi:  0.670nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349569(US10207991, Ex. Cpd. No. 87 | US10611728, Example ...)
Affinity DataKi:  1.10nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349569(US10207991, Ex. Cpd. No. 87 | US10611728, Example ...)
Affinity DataKi:  1.10nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349569(US10207991, Ex. Cpd. No. 87 | US10611728, Example ...)
Affinity DataKi:  1.10nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349570(US10207991, Ex. Cpd. No. 88 | US10611728, Example ...)
Affinity DataKi:  1.30nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349570(US10207991, Ex. Cpd. No. 88 | US10611728, Example ...)
Affinity DataKi:  1.30nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349570(US10207991, Ex. Cpd. No. 88 | US10611728, Example ...)
Affinity DataKi:  1.30nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50232709(CHEMBL4098442 | US11046670, Table 6.3)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50232709(CHEMBL4098442 | US11046670, Table 6.3)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349578(US10207991, Ex. Cpd. No. 103 | US10611728, Example...)
Affinity DataKi:  1.40nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349578(US10207991, Ex. Cpd. No. 103 | US10611728, Example...)
Affinity DataKi:  1.40nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349578(US10207991, Ex. Cpd. No. 103 | US10611728, Example...)
Affinity DataKi:  1.40nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349387(US10207991, Ex. Cpd. No. 18 | US10611728, Example ...)
Affinity DataKi:  1.5nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349387(US10207991, Ex. Cpd. No. 18 | US10611728, Example ...)
Affinity DataKi:  1.5nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349387(US10207991, Ex. Cpd. No. 18 | US10611728, Example ...)
Affinity DataKi:  1.5nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM85609((R)-1-(2-(1-(3-methoxy-benzenesulfonyl)-pyrrolidin...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349577(US10207991, Ex. Cpd. No. 102 | US10611728, Example...)
Affinity DataKi:  1.80nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349478(US10207991, Ex. Cpd. No. 19 | US10611728, Example ...)
Affinity DataKi:  1.80nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349577(US10207991, Ex. Cpd. No. 102 | US10611728, Example...)
Affinity DataKi:  1.80nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349577(US10207991, Ex. Cpd. No. 102 | US10611728, Example...)
Affinity DataKi:  1.80nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349478(US10207991, Ex. Cpd. No. 19 | US10611728, Example ...)
Affinity DataKi:  1.80nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM350897(US9796672, Example Compound 19)
Affinity DataKi:  1.80nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50055523(CHEMBL3321792)
Affinity DataKi:  2.10nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50523091(CHEMBL4577233)
Affinity DataKi:  2.20nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349307(US10207991, Ex. Cpd. No. 4 | US10611728, Example C...)
Affinity DataKi:  2.20nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349307(US10207991, Ex. Cpd. No. 4 | US10611728, Example C...)
Affinity DataKi:  2.20nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50055523(CHEMBL3321792)
Affinity DataKi:  2.20nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50523091(CHEMBL4577233)
Affinity DataKi:  2.20nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349307(US10207991, Ex. Cpd. No. 4 | US10611728, Example C...)
Affinity DataKi:  2.20nMAssay Description:The affinity of candidate sigma-2 ligand compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50232706(CHEMBL4068690 | US11046670, Table 6.2)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50232706(CHEMBL4068690 | US11046670, Table 6.2)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-DTG from the Sigma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50523093(CHEMBL4446729)
Affinity DataKi:  2.5nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349551(US10207991, Ex. Cpd. No. 66 | US10611728, Example ...)
Affinity DataKi:  2.60nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349559(US10207991, Ex. Cpd. No. 76 | US10611728, Example ...)
Affinity DataKi:  2.60nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349559(US10207991, Ex. Cpd. No. 76 | US10611728, Example ...)
Affinity DataKi:  2.60nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM349551(US10207991, Ex. Cpd. No. 66 | US10611728, Example ...)
Affinity DataKi:  2.60nMAssay Description:Radioligand binding assays for Sigma-1 receptors and Sigma-2 receptors were carried out by a commercial contract research organization. For Sigma-1 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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