TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.182nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.204nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.347nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.692nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 0.912nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]RX 821002 from human recombinant adrenergic alpha-2B receptor expressed in CHO cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 1.91nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro binding affinity towards human alpha-2B adrenergic receptor using [3H]-rauwolscineMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity towards human Alpha-2B adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 2.82nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of [3H]- rauwolscine binding to alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibition of [3H]rauwolscine binding to CHO cells expressing the human Alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Inhibition of [3H]rauwolscine binding to CHO cells expressing the human Alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]rauwolscine binding to CHO cells expressing the human Alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Antagonist activity at human recombinant adrenergic alpha2B receptor expressed in CHO cells assessed as inhibition of NE-induced calcium mobilization...More data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL