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Found 579 Enz. Inhib. hit(s) with Target = 'G protein-coupled receptor'
TargetG protein-coupled receptor 34b(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34b(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 119(Canis lupus familiaris)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106206(CHEMBL3598099)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at canine GPR119 by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34b(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560840(CHEMBL4753103)
Affinity DataEC50:  11nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34b(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560840(CHEMBL4753103)
Affinity DataEC50:  12nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM14363(3-(2-propoxyphenyl)-2,4,7,8,9-pentazabicyclo[4.3.0...)
Affinity DataEC50:  61nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 119(Macaca fascicularis)
Amgen

Curated by ChEMBL
LigandPNGBDBM50445481(CHEMBL3104879)
Affinity DataEC50:  73nMAssay Description:Agonist activity at cynomolgus monkey GPR119 assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50323686(Pemirolast)
Affinity DataEC50:  95nMAssay Description:Agonist activity at recombinant rat N-terminal FLAG/eYFP-fused GPR35 expressed in HEK293 cells assessed as induction of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34a(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  129nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34a(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  130nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM78940(METHIOTHEPIN | MLS000859918 | Methiothepin mesylat...)
Affinity DataEC50:  330nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM78940(METHIOTHEPIN | MLS000859918 | Methiothepin mesylat...)
Affinity DataEC50:  331nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34a(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560840(CHEMBL4753103)
Affinity DataEC50:  510nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34a(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560840(CHEMBL4753103)
Affinity DataEC50:  513nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50497861(CHEMBL1824270)
Affinity DataEC50:  930nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50497861(CHEMBL1824270)
Affinity DataEC50:  933nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50404862(CROMOLYN SODIUM | Crolom | Cromoglicic Acid | Crom...)
Affinity DataEC50:  986nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50435998(CHEMBL2392183)
Affinity DataEC50:  991nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436005(CHEMBL2392176)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34b(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34b(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436026(CHEMBL2392148)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436004(CHEMBL2392177)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436019(CHEMBL2392175)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436001(CHEMBL2392174 | CHEMBL2425818)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50435999(CHEMBL2392182)
Affinity DataEC50:  1.54E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436014(CHEMBL2392162)
Affinity DataEC50:  1.76E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436007(CHEMBL2392167)
Affinity DataEC50:  1.83E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436011(CHEMBL2392178)
Affinity DataEC50:  2.05E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436013(CHEMBL2392169)
Affinity DataEC50:  2.08E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436023(CHEMBL2392165)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436009(CHEMBL2392157)
Affinity DataEC50:  2.16E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436020(CHEMBL2392173)
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50497860(CHEMBL1824275)
Affinity DataEC50:  2.50E+3nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50497860(CHEMBL1824275)
Affinity DataEC50:  2.57E+3nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436015(CHEMBL2392161)
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436025(CHEMBL2392153)
Affinity DataEC50:  2.75E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436021(CHEMBL2392168)
Affinity DataEC50:  2.75E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436024(CHEMBL2392164)
Affinity DataEC50:  2.84E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34a(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50497862(CHEMBL1824272)
Affinity DataEC50:  3.09E+3nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor(Human cytomegalovirus)
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50497862(CHEMBL1824272)
Affinity DataEC50:  3.10E+3nMAssay Description:Allosteric modulatory activity at FLAG-tagged human cytomegalovirus US28 receptor delta300 mutant expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436016(CHEMBL2392159)
Affinity DataEC50:  3.13E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436022(CHEMBL2392166)
Affinity DataEC50:  3.14E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor 34a(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436003(CHEMBL2392172)
Affinity DataEC50:  3.25E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436018(CHEMBL2392181)
Affinity DataEC50:  3.61E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436000(CHEMBL2392179)
Affinity DataEC50:  4.17E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436027(CHEMBL2392147)
Affinity DataEC50:  6.65E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor GPR35(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50436010(CHEMBL2392141)
Affinity DataEC50:  8.00E+3nMAssay Description:Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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