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Found 92 Enz. Inhib. hit(s) with Target = 'Glucagon-like peptide 2 receptor'
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183655(CHEMBL3823133)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183893(CHEMBL3823976)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183657(CHEMBL3823541)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183894(CHEMBL3822928)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Rattus norvegicus)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183657(CHEMBL3823541)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at rat GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183892(CHEMBL3822792)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183654(CHEMBL3823835)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183755(CHEMBL3823847)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183756(CHEMBL3823327)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183658(CHEMBL3822459)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183867(CHEMBL3823985)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183659(CHEMBL3824232)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50398387(CHEMBL2177395)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183660(CHEMBL3824079)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183653(CHEMBL3823334)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183650(CHEMBL3823421)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183648(CHEMBL3822888)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Rattus norvegicus)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183895(ALX-0600 | CHEBI:72305 | Gattex Kit | Teduglutide ...)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at rat GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183651(CHEMBL3824241)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183652(CHEMBL3823291)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184061(CHEMBL3823221)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184058(CHEMBL3823876)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184057(CHEMBL3823448)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183895(ALX-0600 | CHEBI:72305 | Gattex Kit | Teduglutide ...)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183661(CHEMBL3823043)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50519608(CHEMBL4534113)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP-2 receptor expressed in CHO-K1 cells assessed as cAMP induction by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183649(CHEMBL3823722)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50398387(CHEMBL2177395)
Affinity DataEC50:  0.0970nMAssay Description:Positive ago-allosteric modulation of GLP2R overexpressed in human SE302 cells assessed as placental alkaline phosphatase activation measured on day ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183574(CHEMBL3822727)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183575(CHEMBL3823786)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183891(CHEMBL3823144)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184066(CHEMBL3824159)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184059(CHEMBL3823889)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183577(CHEMBL3822636)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183642(CHEMBL3823126)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184302(CHEMBL3823411)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184304(CHEMBL3822975)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184307(CHEMBL3823878)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183645(CHEMBL3823818)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183580(CHEMBL3824272)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183672(CHEMBL3824332)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183576(CHEMBL3823643)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183646(CHEMBL3823994)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184315(CHEMBL3822593)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184309(CHEMBL3823333)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183949(CHEMBL3822814)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184055(CHEMBL3822569)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184305(CHEMBL3823755)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50184063(CHEMBL3823051)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 2 receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50183644(CHEMBL3823936)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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