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Found 908 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 4'
LigandPNGBDBM50545036(CHEMBL4632531)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at mouse TRPV4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525957(CHEMBL4461515)
Affinity DataEC50:  49nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525953(CHEMBL4437589)
Affinity DataEC50:  60nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
LigandPNGBDBM50277487(4alpha-Phorbol 12,13-dihexanoate | CHEMBL490470)
Affinity DataEC50:  70nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525945(CHEMBL4449495)
Affinity DataEC50:  125nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50545034(CHEBI:34450 | CHEMBL1893588)
Affinity DataEC50:  150nMAssay Description:Agonist activity at mouse TRPV4More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50277491(CHEMBL504955 | Lumi-4alpha-Phorbol 12,13-didecanoa...)
Affinity DataEC50:  175nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525954(CHEMBL4474443)
Affinity DataEC50:  200nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525947(CHEMBL4560730)
Affinity DataEC50:  280nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50240777(4alpha-phorbol-didecanoate | CHEMBL118987 | Decano...)
Affinity DataEC50:  370nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
LigandPNGBDBM50240777(4alpha-phorbol-didecanoate | CHEMBL118987 | Decano...)
Affinity DataEC50:  370nMAssay Description:Agonist activity at mouse TRPV4More data for this Ligand-Target Pair
LigandPNGBDBM50277486(4alpha-Phorbol 13-decanoate | CHEMBL541720)
Affinity DataEC50:  450nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50318486(2-Methyl-2-(4-methyl-pent-3-enyl)-7-pentyl-2H-chro...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525942(CHEMBL4465567)
Affinity DataEC50:  663nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525952(CHEMBL4542977)
Affinity DataEC50:  670nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525944(CHEMBL4585693)
Affinity DataEC50:  740nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50426574(CHEMBL2324348)
Affinity DataEC50:  770nMAssay Description:Agonist activity at TRPV4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50545035(CHEMBL4303584)
Affinity DataEC50:  770nMAssay Description:Agonist activity at mouse TRPV4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525955(CHEMBL4455286)
Affinity DataEC50:  870nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50532215(CBD-V | CBDV | Cannabidivarin | GWP42006)
Affinity DataEC50:  900nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50318484(2-((1R,6R)-6-Isopropenyl-3-methyl-cyclohex-2-enyl)...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at rat TRPV4 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525948(CHEMBL4516018)
Affinity DataEC50:  910nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525960(CHEMBL4440011)
Affinity DataEC50:  920nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525958(CHEMBL4591600)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525959(CHEMBL4454987)
Affinity DataEC50:  1.44E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525946(CHEMBL4586856)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50277490(4alpha-Phorbol 12,13-dimyristate | CHEMBL451849)
Affinity DataEC50:  2.83E+3nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525943(CHEMBL4449850)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50548384(CHEMBL4762439)
Affinity DataEC50:  6.20E+3nMAssay Description:Agonist activity at rat TRPV4 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye bas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50511105(GWP-42004 | Gwp42004 | O-4394 | THCV | Tetrahydroc...)
Affinity DataEC50:  6.40E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50285610(CBV | CHEMBL4170268)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50285610(CBV | CHEMBL4170268)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525949(CHEMBL4436655)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525956(CHEMBL4465513)
Affinity DataEC50:  1.22E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50571573(CHEMBL4863993)
Affinity DataEC50: <1.58E+4nMAssay Description:Agonist activity at human TRPV4 expressed in HEK cells assessed as increase in GSK1016790A-induced intracellular calcium level measured after 1 hr by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50602168(CHEMBL5192928)
Affinity DataEC50: <1.58E+4nMAssay Description:Agonist activity at human TRPV4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50571572(CHEMBL4854482)
Affinity DataEC50: <1.58E+4nMAssay Description:Agonist activity at human TRPV4 expressed in HEK cells assessed as increase in GSK1016790A-induced intracellular calcium level measured after 1 hr by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50571570(CHEMBL4876211)
Affinity DataEC50: <1.58E+4nMAssay Description:Agonist activity at human TRPV4 expressed in HEK cells assessed as increase in GSK1016790A-induced intracellular calcium level measured after 1 hr by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50571571(CHEMBL4849726)
Affinity DataEC50: <1.58E+4nMAssay Description:Agonist activity at human TRPV4 expressed in HEK cells assessed as increase in GSK1016790A-induced intracellular calcium level measured after 1 hr by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol |...)
Affinity DataEC50:  1.61E+4nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol |...)
Affinity DataEC50:  1.61E+4nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50463443(CHEMBL4241477)
Affinity DataEC50:  1.80E+4nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataEC50:  2.25E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525950(CHEMBL4552995)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525951(CHEMBL4447367)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50277740(4-Deoxy-4alpha-Phorbol 12,13-didecanoate | CHEMBL5...)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50277739(4alpha-phorbol diacetate | CHEMBL484343)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50277488(4alpha-Phorbol 12,13-dioctanoate | CHEMBL507303)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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