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Found 420 Enz. Inhib. hit(s) with Target = 'Acetylcholine receptor'
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023330(1-(9-Aza-bicyclo[4.2.1]non-2-en-2-yl)-ethanone | 1...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023331((+)-pyrido[3,4-b]homotropane | (+/-)-pyrido[3,4-b]...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of [3H]-MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit delta(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50547502(CHEMBL4793300)
Affinity DataIC50:  0.184nMAssay Description:Inhibition of rat alpha1beta1epsilondelta expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current respons...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487992(CHEMBL2270633)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023331((+)-pyrido[3,4-b]homotropane | (+/-)-pyrido[3,4-b]...)
Affinity DataIC50:  1nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023330(1-(9-Aza-bicyclo[4.2.1]non-2-en-2-yl)-ethanone | 1...)
Affinity DataIC50:  1nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50486231(CHEBI:39177 | CLOTHIANIDINE)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50486231(CHEBI:39177 | CLOTHIANIDINE)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596365(CHEMBL5179810)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50251868((Z)-thiacloprid | CHEMBL451432 | {(2Z)-3-[(6-chlor...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit gamma(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50547502(CHEMBL4793300)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of rat (alpha1)2betagammadelta expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current respons...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50:  4nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487983(CHEMBL148390)
Affinity DataIC50:  4.40nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516960(CHEMBL4435544)
Affinity DataIC50:  6nMAssay Description:Inhibition of AChE (unknown origin) after 2 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50547500(CHEMBL4759352)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of rat (alpha1)2betagammadelta expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current respons...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487983(CHEMBL148390)
Affinity DataIC50:  7.40nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50251868((Z)-thiacloprid | CHEMBL451432 | {(2Z)-3-[(6-chlor...)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit gamma(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50547501(CHEMBL4788244)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of rat (alpha1)2betagammadelta expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current respons...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487979(IMIDACLOTHIZ)
Affinity DataIC50:  8.20nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50486223(CHEBI:39164 | acetamiprid)
Affinity DataIC50:  8.30nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit gamma(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50547503(CHEMBL4753712)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of rat (alpha1)2betagammadelta expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current respons...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487980(DESMETHYLTHIAMETHOXAM)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50486236(CHEBI:39170 | NITENPYRAM)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596366(CHEMBL5204683)
Affinity DataIC50:  12nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487985(CHEMBL2269823)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487979(IMIDACLOTHIZ)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487980(DESMETHYLTHIAMETHOXAM)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50487985(CHEMBL2269823)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516959(CHEMBL4471876)
Affinity DataIC50:  27nMAssay Description:Inhibition of AChE (unknown origin) after 2 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596377(CHEMBL5181578)
Affinity DataIC50:  32nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596341(CHEMBL5176418)
Affinity DataIC50:  36nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  44nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596380(CHEMBL5173121)
Affinity DataIC50:  44nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516976(CHEMBL4518438)
Affinity DataIC50:  47nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50459975(CHEMBL4228909)
Affinity DataIC50:  50nMAssay Description:Inhibition of nAChR epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516974(CHEMBL4516351)
Affinity DataIC50:  57nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516977(CHEMBL4518992)
Affinity DataIC50:  58nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596378(CHEMBL5207035)
Affinity DataIC50:  58nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516975(CHEMBL4514263)
Affinity DataIC50:  62nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596367(CHEMBL5190924)
Affinity DataIC50:  71nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516963(CHEMBL2376519)
Affinity DataIC50:  82nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596382(CHEMBL5188135)
Affinity DataIC50:  83nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596360(CHEMBL5200573)
Affinity DataIC50:  87nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50516982(CHEMBL4447626)
Affinity DataIC50:  88nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50596381(CHEMBL5179648)
Affinity DataIC50:  91nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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