Compile Data Set for Download or QSAR
maximum 50k data
Found 7016 Enz. Inhib. hit(s) with Target = 'Apelin receptor'
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078007(CHEMBL3417384)
Affinity DataIC50:  0.0200nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataIC50:  0.0250nMAssay Description:Displacement of [125I]-(Glp1,Nle11,Try14)apelin-13 from recombinant rat EGFP-fused apelin receptor expressed in CHO cell membrane measured after 3 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554009(CHEMBL4787992)
Affinity DataIC50:  0.0501nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554014(CHEMBL4751860)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554012(CHEMBL4764067)
Affinity DataIC50:  0.219nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077994(CHEMBL3417378)
Affinity DataIC50:  0.25nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554013(CHEMBL4786278)
Affinity DataIC50:  0.295nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554010(CHEMBL4795982)
Affinity DataIC50:  0.302nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554011(CHEMBL4750105)
Affinity DataIC50:  0.302nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078002(CHEMBL3417389)
Affinity DataIC50:  0.430nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078006(CHEMBL3417385)
Affinity DataIC50:  0.480nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554001(CHEMBL4789383)
Affinity DataIC50:  0.550nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077995(CHEMBL3417377)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50257231(CHEMBL4065973)
Affinity DataIC50:  0.603nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078001(CHEMBL3417390)
Affinity DataIC50:  0.860nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554007(CHEMBL4740668)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553994(CHEMBL4753692)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553993(CHEMBL4744011)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553999(CHEMBL4759447)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077993(CHEMBL3417379)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553992(CHEMBL4797426)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078005(CHEMBL3417386)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554008(CHEMBL4758442)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077992(CHEMBL3417380)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554003(CHEMBL4755954)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554002(CHEMBL4775988)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553998(CHEMBL4788623)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078000(CHEMBL3414601)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554000(CHEMBL4799454)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553995(CHEMBL4761000)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583256(CHEMBL5087847)
Affinity DataIC50:  2.20nMAssay Description:Inhibition [125I]-[Nle75,Tyr77][Pyr1]-Ape13 binding to YFP-tagged human wildtype APJ expressed in HEK293 cell membranes incubated for 1 hr by scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553991(CHEMBL4745212)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553997(CHEMBL4763310)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554006(CHEMBL4744024)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077999(CHEMBL3417291)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078003(CHEMBL3417388)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50553996(CHEMBL4794535)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554005(CHEMBL4741692)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583256(CHEMBL5087847)
Affinity DataIC50:  5.40nMAssay Description:Inhibition [125I]-[Nle75,Tyr77][Pyr1]-Ape13 binding to YFP-tagged human APJ E20A mutant expressed in HEK293 cell membranes incubated for 1 hr by scin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078010(CHEMBL3417381)
Affinity DataIC50:  6.10nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554004(CHEMBL4760648)
Affinity DataIC50:  6.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078008(CHEMBL3417383)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077997(CHEMBL3417375)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077998(CHEMBL3414600)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078004(CHEMBL3417387)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078009(CHEMBL3417382)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583262(CHEMBL5079665)
Affinity DataIC50:  15nMAssay Description:Inhibition [125I]-[Nle75,Tyr77][Pyr1]-Ape13 binding to YFP-tagged human wildtype APJ expressed in HEK293 cell membranes incubated for 1 hr by scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583256(CHEMBL5087847)
Affinity DataIC50:  17nMAssay Description:Inhibition [125I]-[Nle75,Tyr77][Pyr1]-Ape13 binding to YFP-tagged human APJ D32A mutant expressed in HEK293 cell membranes incubated for 1 hr by scin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50077996(CHEMBL3417376)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]apelin-13[Glp65,Nle75,Tyr77] from YFP epitope-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 7016 total ) | Next | Last >>
Jump to: