Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of rat epididymis beta-mannosidase by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+4nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of rat epididymis beta-mannosidase by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+5nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+5nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+5nMAssay Description:Inhibition of rat epididymis beta-mannosidase assessed as p-nitrophenol release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+5nMAssay Description:Inhibition of rat epididymis beta-mannosidase by spectrophotometryMore data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:The compound was tested for its inhibitory activity against beta-mannosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 57nM ΔG°: -43.0kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 72nM ΔG°: -42.4kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 401nM ΔG°: -38.0kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 975nM ΔG°: -35.7kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nM ΔG°: -35.6kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nM ΔG°: -34.8kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nM ΔG°: -34.0kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nM ΔG°: -33.7kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nM ΔG°: -33.7kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nM ΔG°: -33.6kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nM ΔG°: -33.4kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition against Beta-mannosidase in snailMore data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:The compound was tested for its inhibitory activity against beta-mannosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nM ΔG°: -29.4kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nM ΔG°: -29.0kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:The compound was tested for its inhibitory activity against beta-mannosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+4nM ΔG°: -27.7kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition against Beta-mannosidase in snailMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+5nM ΔG°: -19.6kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nM ΔG°: -17.8kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+6nM ΔG°: -16.0kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+6nM ΔG°: -13.2kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 9.00E+6nM ΔG°: -12.1kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+7nM ΔG°: -11.6kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+7nM ΔG°: -11.0kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+7nM ΔG°: -10.1kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.30E+7nM ΔG°: -9.73kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+7nM ΔG°: -8.80kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: >4.00E+8nM ΔG°: >-2.36kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair