Found 562 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' 
Affinity DataIC50: 0.0820nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMpH: 7.3 T: 2°CAssay Description:Membranes were incubated with [125I] kisspeptin-15 and increasing concentrations of test compound in binding buffer. The reaction mixtures were dilut...More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Displacement of [125I]kisspeptin-15 from GPR54More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMpH: 7.3 T: 2°CAssay Description:Membranes were incubated with [125I] kisspeptin-15 and increasing concentrations of test compound in binding buffer. The reaction mixtures were dilut...More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Displacement of [125I]kisspeptin-15 from GPR54More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMpH: 7.3 T: 2°CAssay Description:Membranes were incubated with [125I] kisspeptin-15 and increasing concentrations of test compound in binding buffer. The reaction mixtures were dilut...More data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.610nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMpH: 7.3 T: 2°CAssay Description:Membranes were incubated with [125I] kisspeptin-15 and increasing concentrations of test compound in binding buffer. The reaction mixtures were dilut...More data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:Displacement of [125I]kisspeptin-15 from GPR54More data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Affinity DataIC50: 0.830nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMpH: 7.3 T: 2°CAssay Description:Membranes were incubated with [125I] kisspeptin-15 and increasing concentrations of test compound in binding buffer. The reaction mixtures were dilut...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]metastin from human GPR54 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]metastin from human GPR54 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]metastin(40-54) from human GPR54 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Displacement of [125I]metastin from human GPR54 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Displacement of [125I]metastin from human GPR54 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMpH: 7.3 T: 2°CAssay Description:Membranes were incubated with [125I] kisspeptin-15 and increasing concentrations of test compound in binding buffer. The reaction mixtures were dilut...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
