TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 20.4nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 20.8nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 23nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 26nMAssay Description:Inhibition of Orai1 (unknown origin) by patch clamp assayMore data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 32.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 34.1nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 35.7nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 36.4nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 37.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 39.2nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 47.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 48nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 48.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 48.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 50.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 51.3nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 52.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 53.4nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 60nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 60.3nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 62.4nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 62.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 63.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 65.5nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 70.3nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 72nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 72.1nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein/Stromal interaction molecule 1(Homo sapiens (Human))
Lupin
Curated by ChEMBL
Lupin
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of Orai1/STIM1 (unknown origin) expressed in HEK293 cells assessed as reduction in Ca2+-release activated Ca2+ entry current by manual pat...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 81.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 86.1nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 98.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 99.7nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: <100nMAssay Description:Inhibition of human Orai1/STIM1 expressed in HEK293 cells assessed as inhibition of channel-mediated calcium current by electrophysiology assay in pr...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 104nMAssay Description:Inhibition of human Orai1/STIM1 expressed in HEK293 cells assessed as inhibition of channel-mediated calcium current by electrophysiology assay in pr...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein/Stromal interaction molecule 1(Homo sapiens (Human))
Lupin
Curated by ChEMBL
Lupin
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of Orai1/STIM1 (unknown origin)More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 120nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 124nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 124nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 130nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 139nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataIC50: 141nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair