Compile Data Set for Download or QSAR
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Found 332 Enz. Inhib. hit(s) with Target = 'Protein kinase C gamma'
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327943(Aplysiatoxin | CHEMBL1256416)
Affinity DataKi:  0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50587724(CHEMBL5175742)
Affinity DataKi:  0.650nMAssay Description:Displacement of 3H-PDBu from recombinant human PKCgamma incubated for 25 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057514((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-5...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human Protein kinase C gamma with [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  1.60nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50097750(Butyric acid (1aR,1bS,4aS,7aR,7bR,8R,9R,9aS)-9-but...)
Affinity DataKi:  1.80nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]- PDBu binding to peptide C, rat brain PKC gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  2.90nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)
Affinity DataKi:  4.90nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50097750(Butyric acid (1aR,1bS,4aS,7aR,7bR,8R,9R,9aS)-9-but...)
Affinity DataKi:  5.20nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  5.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  19.4nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataKi:  22nMAssay Description:Displacement of 3H-PDBu from recombinant human PKCgamma incubated for 25 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  39nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  39nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  40.7nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  43nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  53nMAssay Description:Inhibition of [3H]- PDBu binding to peptide C, rat brain PKC gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50374190(CHEMBL271403)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327944((1S,3R,5R,9R,13R)-9-Hydroxymethyl-16,16-dimethyl-3...)
Affinity DataKi:  80nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  138nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  151nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50099064(CHEMBL368720 | Dodecanoic acid (3S,3aR,8R,8aS)-3-h...)
Affinity DataKi:  209nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50463479(CHEMBL4249925)
Affinity DataKi:  210nMAssay Description:Inhibition of PKCgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  213nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1b domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  213nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50374190(CHEMBL271403)
Affinity DataKi:  225nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50374191(CHEMBL261387)
Affinity DataKi:  234nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50099065((3S,3aR,8R,8aS)-6-Dec-1-ynyl-3-hydroxymethyl-8-iso...)
Affinity DataKi:  279nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50092015((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3...)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50092015((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3...)
Affinity DataKi:  296nMAssay Description:Binding affinity for Protein kinase C beta C1b domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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