TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: >6.71E+3nMAssay Description:Inhibition of NEK4More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of full-length recombinant human GST-tagged NEK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 74.2nMAssay Description:Inhibition of human NEK4 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of human NEK4 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of full-length recombinant human GST-tagged NEK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of full-length recombinant human GST-tagged NEK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of full-length recombinant human GST-tagged NEK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of NEK4More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length GST-tagged NEK4 expressed in baculovirus expression systemMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human NEK4 using MBP as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full-length human NEK4 P225A mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NEK4 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant full length human GST-tagged NEK4 expressed in baculovirus expression system using serine/threonine-7 peptide as substrate ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for NEK4 kinase domainMore data for this Ligand-Target Pair