Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'ADP-ribose glycohydrolase MACROD2'
TargetADP-ribose glycohydrolase MACROD2(Homo sapiens)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50460478(CHEMBL4226903)
Affinity DataKd:  150nMAssay Description:Binding affinity to human MDO2 by ITCMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetADP-ribose glycohydrolase MACROD2(Homo sapiens)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50595207(CHEMBL5208626)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of N-terminal His-TEV-V5 tagged human Mdo2 (7 to 243 residues) expressed in Escherichia coli BL21 (DE3) using BIO-6His tagged linker pepti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetADP-ribose glycohydrolase MACROD2(Homo sapiens)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50088433(Dihydralazine)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of human Mdo2More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetADP-ribose glycohydrolase MACROD2(Homo sapiens)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50595206(CHEMBL5205107)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of N-terminal His-TEV-V5 tagged human Mdo2 (7 to 243 residues) expressed in Escherichia coli BL21 (DE3) using BIO-6His tagged linker pepti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed