TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 0.0900nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 0.0930nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.0930nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.100nMAssay Description:Binding affinity to human EPHA3More data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.80nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 8.60nMAssay Description:Binding affinity to EphA3 (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 27nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 27nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
Affinity DataKd: 39.3nMAssay Description:Binding affinity to EphA3 (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding affinity to human EPHA3More data for this Ligand-Target Pair
Affinity DataKd: 55nMAssay Description:Average Binding Constant for EPHA3; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 80nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity to EPHA3More data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Inhibition of EPHA3 (unknown origin) assessed as dissociation constant by ELISA-like binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 360nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 390nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 580nMAssay Description:Average Binding Constant for EPHA3; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Average Binding Constant for EPHA3; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 700nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 747nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged EPHA3 (unknown origin) (579 to 983 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair
Affinity DataKd: 810nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 880nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 880nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 880nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 1.50E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity to N-terminal His tagged EphA3 LBD (unknown origin) expressed in Rosetta-Gami B(DE3) cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Average Binding Constant for EPHA3; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding affinity to EPHA3More data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 1.90E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 2.00E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.10E+3nMAssay Description:Binding affinity to EPHA3More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 2.10E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 2.10E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3 [1-975](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 2.10E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 2.10E+3nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair