Found 79 Enz. Inhib. hit(s) with Target = 'Microtubule-associated serine/threonine-protein kinase 1'
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 40nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 350nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 520nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 3.30E+3nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 4.60E+3nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 5.50E+3nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 6.20E+3nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAST1More data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair
TargetMicrotubule-associated serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAST1 kinase domainMore data for this Ligand-Target Pair