Affinity DataKd: 0.300nMAssay Description:Kinase binding assays were performed at DiscoveRx using the general KINOMEscan Kd Protocol (Fabian, M. A. et al., “A small molecule-kinase interactio...More data for this Ligand-Target Pair
Affinity DataKd: 0.300nMAssay Description:Kinase binding assays were performed at DiscoveRx using the general KINOMEscan Kd Protocol (Fabian, M. A. et al., “A small molecule-kinase interactio...More data for this Ligand-Target Pair
Affinity DataKd: 3.40nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 4.90nMAssay Description:Binding affinity to wild-type human partial length TRKC (Q531 to G825 residues) expressed in mammalian expression system by Kinomescan method relativ...More data for this Ligand-Target Pair
Affinity DataKd: 9.30nMAssay Description:Binding affinity to human TrkCMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity to TRKCMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Binding affinity to wild type human partial length TRKC (531 to 825 residues) expressed in mammalian expression system preincubated for 1 hr measured...More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Binding affinity to TrkC (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Binding affinity to wild type human partial length TRKC (531 to 825 residues) expressed in mammalian expression system preincubated for 1 hr measured...More data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged NTRK3 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair
Affinity DataKd: 23nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged NTRK3 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 68nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 82nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:Binding affinity to TRKCMore data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 570nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding affinity to TRKCMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 930nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for TRKC kinase domainMore data for this Ligand-Target Pair