Compile Data Set for Download or QSAR
maximum 50k data
Found 427 Enz. Inhib. hit(s) with Target = 'Protein delta homolog 1'
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50441567(CHEMBL2436978 | US10485800, Example 181)
Affinity DataKd:  70nMAssay Description:Binding affinity to human wild type DLK by qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKd:  100nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  840nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM13535(4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50042942(CHEMBL3355003)
Affinity DataKi:  0.170nMAssay Description:Inhibition of DLK (unknown origin) by RT-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50042940(CHEMBL3355005)
Affinity DataKi:  0.400nMAssay Description:Inhibition of DLK (unknown origin) by RT-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  36nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50042941(CHEMBL3355004)
Affinity DataKi:  110nMAssay Description:Inhibition of DLK (unknown origin) by RT-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50042939(CHEMBL3355006)
Affinity DataKi:  270nMAssay Description:Inhibition of DLK (unknown origin) by RT-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50441567(CHEMBL2436978 | US10485800, Example 181)
Affinity DataIC50:  150nMAssay Description:Inhibition of human wild type DLK by qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50429477(CHEMBL2332840)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50458548(CHEMBL4218417)
Affinity DataIC50:  119nMAssay Description:Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM50458549(CHEMBL4207983)
Affinity DataIC50:  1nMAssay Description:Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
Affinity DataIC50:  114nMAssay Description:Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637456(US20230382904, Compound 371)
Affinity DataIC50:  500nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637457(US20230382904, Compound 372)
Affinity DataIC50:  430nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637458(US20230382904, Compound 373)
Affinity DataIC50:  370nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637459(US20230382904, Compound 374)
Affinity DataIC50:  280nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637460(US20230382904, Compound 375)
Affinity DataIC50:  840nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637461(US20230382904, Compound 376)
Affinity DataIC50:  260nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637462(US20230382904, Compound 377)
Affinity DataIC50:  210nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637463(US20230382904, Compound 378)
Affinity DataIC50:  1.80E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637464(US20230382904, Compound 379)
Affinity DataIC50:  970nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637465(US20230382904, Compound 380)
Affinity DataIC50:  1.10E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637466(US20230382904, Compound 381)
Affinity DataIC50:  380nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637467(US20230382904, Compound 382)
Affinity DataIC50:  310nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637468(US20230382904, Compound 383)
Affinity DataIC50: >3.00E+4nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637469(US20230382904, Compound 384)
Affinity DataIC50: >3.00E+4nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637470(US20230382904, Compound 385)
Affinity DataIC50:  1.10E+4nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637471(US20230382904, Compound 386)
Affinity DataIC50:  3.40E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637472(US20230382904, Compound 387)
Affinity DataIC50:  750nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637473(US20230382904, Compound 388)
Affinity DataIC50:  210nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637474(US20230382904, Compound 389)
Affinity DataIC50: >3.00E+4nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637475(US20230382904, Compound 390)
Affinity DataIC50:  1.10E+4nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637476(US20230382904, Compound 391)
Affinity DataIC50:  2.00E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637477(US20230382904, Compound 392)
Affinity DataIC50:  100nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637478(US20230382904, Compound 393)
Affinity DataIC50:  260nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637479(US20230382904, Compound 394)
Affinity DataIC50:  410nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637480(US20230382904, Compound 395)
Affinity DataIC50:  1.10E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637481(US20230382904, Compound 396)
Affinity DataIC50:  310nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637482(US20230382904, Compound 397)
Affinity DataIC50:  73nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637483(US20230382904, Compound 398)
Affinity DataIC50:  880nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637484(US20230382904, Compound 399)
Affinity DataIC50:  1.76E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637485(US20230382904, Compound 400)
Affinity DataIC50:  2.15E+3nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein delta homolog 1(Homo sapiens (Human))
Califia Bio

Curated by ChEMBL
LigandPNGBDBM637486(US20230382904, Compound 401)
Affinity DataIC50:  8.10nMAssay Description:Assay Protocol for 1536 MTP format: test compounds were predispensed (60 nl) in test plates; +3 μl DLK solution (10 nM DLK, catalytic domain, Ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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