Affinity DataKd: 0.800nMAssay Description:Binding affinity to human ESD expressed in HEK293T cells assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Binding affinity to human ESD expressed in HEK293T cells assessed as dissociation rate constantMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Tested for inhibition of substrate hydrolysis in the presence of porcine kidney esterase at a concentration of 10 nMMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:pA2 value towards endothelin receptor A was determined as functional ETA antagonismMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Tested for inhibition of substrate hydrolysis in the presence of porcine kidney esterase at a concentration of 9 uMMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:pA2 value towards endothelin receptor A was determined as functional ETA antagonismMore data for this Ligand-Target Pair