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Found 571 Enz. Inhib. hit(s) with Target = 'Galectin-1'
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21519(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-(carbam...)
Affinity DataKd:  4.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21521(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  4.90E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21522(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  3.40E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21523(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(butyl...)
Affinity DataKd:  2.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21524(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(dieth...)
Affinity DataKd:  4.60E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21525(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  4.90E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21533(N-[(2R,3R,4R,5S,6R)-4-hydroxy-6-(hydroxymethyl)-2-...)
Affinity DataKd:  7.00E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21527(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  4.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21528(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(benzy...)
Affinity DataKd:  3.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21529(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  4.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21530(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(cyclo...)
Affinity DataKd:  4.00E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21531(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  1.60E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21532(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-({[(2S,...)
Affinity DataKd:  5.80E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21526(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  2.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120768(US8703720, Reference Compound 1)
Affinity DataKd: >1.00E+7nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120769(US8703720, Reference Compound 2)
Affinity DataKd:  6.50E+4nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120771(US8703720, 15)
Affinity DataKd:  1.90E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120772(US8703720, 16)
Affinity DataKd:  1.50E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120773(US8703720, 17)
Affinity DataKd:  1.20E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120774(US8703720, 18)
Affinity DataKd:  350nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120775(US8703720, 19)
Affinity DataKd:  1.30E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM120776(US8703720, 23)
Affinity DataKd:  6.30E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-1 [C3S](Homo sapiens (Human))
Universit?? De Nantes

LigandPNGBDBM223990(2-[6-Maleimide)caproyl]ethyl [3-O-(2-naphthyl)meth...)
Affinity DataKd:  1.60E+4nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-1 [C3S](Homo sapiens (Human))
Universit?? De Nantes

LigandPNGBDBM223990(2-[6-Maleimide)caproyl]ethyl [3-O-(2-naphthyl)meth...)
Affinity DataKd:  4.30E+4nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-1 [C3S](Homo sapiens (Human))
Universit?? De Nantes

LigandPNGBDBM223991([3-O-(2-naphthyl)methyl-β-D-galactopyranosyl]...)
Affinity DataKd:  2.70E+4nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-1 [C3S](Homo sapiens (Human))
Universit?? De Nantes

LigandPNGBDBM223992(4-O-[3-O-(3-methoxybenzyl)-β-D-galactopyranos...)
Affinity DataKd:  2.30E+4nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-1 [C3S](Homo sapiens (Human))
Universit?? De Nantes

LigandPNGBDBM223993(TD139)
Affinity DataKd:  2.20E+3nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048091(CHEMBL3311520)
Affinity DataKd:  3.60E+6nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048092(CHEMBL3311521)
Affinity DataKd:  5.00E+5nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243888(CHEMBL442951 | methyl beta-D-galactopyranoside | m...)
Affinity DataKd:  1.00E+7nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048093(CHEBI:610092 | CHEMBL503075 | Lactoside | Methyl B...)
Affinity DataKd:  1.90E+5nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048094(CHEMBL3311522)
Affinity DataKd:  1.70E+6nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048095(CHEMBL3311523)
Affinity DataKd:  5.10E+6nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048096(CHEMBL3311524)
Affinity DataKd:  6.50E+5nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048097(CHEMBL3311525)
Affinity DataKd:  4.50E+6nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048098(CHEMBL3311526)
Affinity DataKd:  1.90E+6nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM21540(Galactose-Derived Compound 18 | N-[(2R,3R,4S,5R,6S...)
Affinity DataKd:  9.80E+5nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50034081(CHEBI:55507 | CHEMBL467773)
Affinity DataKd: >1.00E+7nMAssay Description:Antagonist activity against human galectin 1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50244378((2R,3S,4S,5S,6R)-3,5-dihydroxy-2-(hydroxymethyl)-6...)
Affinity DataKd:  2.00E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243801(CHEMBL486246 | triethylammonium (2R,3S,4S,5S,6R)-5...)
Affinity DataKd: >4.00E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243734(CHEMBL479534 | triethylazanium (2R,3S,4S,5S,6R)-5-...)
Affinity DataKd:  4.40E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243733(CHEMBL471377 | triethylammonium (2R,3S,4S,5S,6R)-5...)
Affinity DataKd: >4.00E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243732(CHEMBL511306 | triethylammonium (2R,3S,4S,5S,6R)-5...)
Affinity DataKd: >4.00E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243731((2R,3S,4S,5S,6R)-3-acetoxy-5-hydroxy-6-(hydroxymet...)
Affinity DataKd: >4.00E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50244379((2R,3S,4S,5S,6R)-3-hydroxy-2-(hydroxymethyl)-6-met...)
Affinity DataKd:  1.80E+6nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50244377(CHEMBL502337 | methyl beta-D-talopyranoside)
Affinity DataKd: >1.00E+7nMAssay Description:Binding affinity to human galectin1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50420903(CHEMBL221186)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to human [15N]-labelled Galectin-1 by heteronuclear NMR spectroscopy analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50425514(CHEMBL2313334)
Affinity DataKd:  6.70E+3nMAssay Description:Binding affinity to galectin-1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50425515(CHEMBL2313335)
Affinity DataKd:  2.80E+4nMAssay Description:Binding affinity to galectin-1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-1(Homo sapiens (Human))
Lund University

LigandPNGBDBM50425516(CHEMBL2313336)
Affinity DataKd:  1.80E+5nMAssay Description:Binding affinity to galectin-1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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