Compile Data Set for Download or QSAR
maximum 50k data
Found 1474 Enz. Inhib. hit(s) with Target = 'Galectin-3'
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21519(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-(carbam...)
Affinity DataKd:  6.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21521(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  3.80E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21522(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  5.20E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21523(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(butyl...)
Affinity DataKd:  2.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21524(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(dieth...)
Affinity DataKd:  4.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21525(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  7.40E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21526(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  6.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21527(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  4.00E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21528(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(benzy...)
Affinity DataKd:  1.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21529(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  3.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21530(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(cyclo...)
Affinity DataKd:  5.70E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21531(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  6.90E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21532(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-({[(2S,...)
Affinity DataKd:  1.60E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21533(N-[(2R,3R,4R,5S,6R)-4-hydroxy-6-(hydroxymethyl)-2-...)
Affinity DataKd:  6.70E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21534(Galactose-Derived Compound 12 | [(2S,3R,4S,5R,6R)-...)
Affinity DataKd:  8.70E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21535(Galactose-Derived Compound 13 | {[(2S,3R,4S,5R,6R)...)
Affinity DataKd:  1.50E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21536(Galactose-Derived Compound 14 | {[(2S,3R,4S,5R,6R)...)
Affinity DataKd:  2.50E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21537((benzyloxy)({[(2S,3R,4S,5R,6R)-5-hydroxy-6-(hydrox...)
Affinity DataKd:  1.20E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21538((2S,3R,4S,5R,6R)-5-hydroxy-6-(hydroxymethyl)-4-[(4...)
Affinity DataKd:  2.40E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21539(Galactose-Derived Compound 17 | N-[(2S,3R,4S,5R,6R...)
Affinity DataKd:  3.80E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21540(Galactose-Derived Compound 18 | N-[(2R,3R,4S,5R,6S...)
Affinity DataKd:  2.20E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21541((2R,3R,4S,5R,6S)-2-(hydroxymethyl)-6-(methylsulfan...)
Affinity DataKd:  5.90E+6nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM21542(Galactose-Derived Compound 20 | [(2S,3R,4S,5R,6R)-...)
Affinity DataKd:  2.80E+6nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120768(US8703720, Reference Compound 1)
Affinity DataKd:  4.40E+6nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120769(US8703720, Reference Compound 2)
Affinity DataKd:  5.90E+4nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120770(US8703720, 7)
Affinity DataKd:  430nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120771(US8703720, 15)
Affinity DataKd:  230nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120772(US8703720, 16)
Affinity DataKd:  150nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120773(US8703720, 17)
Affinity DataKd:  210nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120774(US8703720, 18)
Affinity DataKd:  550nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120775(US8703720, 19)
Affinity DataKd:  190nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM120776(US8703720, 23)
Affinity DataKd:  1.40E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223990(2-[6-Maleimide)caproyl]ethyl [3-O-(2-naphthyl)meth...)
Affinity DataKd:  14nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223990(2-[6-Maleimide)caproyl]ethyl [3-O-(2-naphthyl)meth...)
Affinity DataKd:  82nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223991([3-O-(2-naphthyl)methyl-β-D-galactopyranosyl]...)
Affinity DataKd:  590nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223991([3-O-(2-naphthyl)methyl-β-D-galactopyranosyl]...)
Affinity DataKd:  2.99E+3nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223992(4-O-[3-O-(3-methoxybenzyl)-β-D-galactopyranos...)
Affinity DataKd:  660nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223992(4-O-[3-O-(3-methoxybenzyl)-β-D-galactopyranos...)
Affinity DataKd:  3.27E+3nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223993(TD139)
Affinity DataKd:  36nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM223993(TD139)
Affinity DataKd:  166nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50336204(12-Mercaptododecyl-beta-D-galactopyranosyl-(1->4)-...)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity to human galectin-3 by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50336202(12-Mercaptododecyl-beta-D-galactopyranosyl-(1->4)-...)
Affinity DataKd:  1.43E+3nMAssay Description:Binding affinity to human galectin-3 by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50336203(12-Mercaptododecyl-beta-D-galactopyranosyl-(1->4)-...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to human galectin-3 by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50370453(LACTOSE | Lactose, anhydrous)
Affinity DataKd:  2.30E+5nMAssay Description:Binding affinity to galectin-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50045334(CHEMBL3337492)
Affinity DataKd:  1.82E+4nMAssay Description:Binding affinity to galectin-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50045335(CHEMBL3337493)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to galectin-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048091(CHEMBL3311520)
Affinity DataKd:  1.00E+7nMAssay Description:Antagonist activity against human galectin 3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048092(CHEMBL3311521)
Affinity DataKd:  1.30E+5nMAssay Description:Antagonist activity against human galectin 3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50243888(CHEMBL442951 | methyl beta-D-galactopyranoside | m...)
Affinity DataKd:  4.40E+6nMAssay Description:Antagonist activity against human galectin 3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-3(Homo sapiens (Human))
Lund University

LigandPNGBDBM50048093(CHEBI:610092 | CHEMBL503075 | Lactoside | Methyl B...)
Affinity DataKd:  2.20E+5nMAssay Description:Antagonist activity against human galectin 3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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