TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKd: 1.20nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKd: 1.12E+3nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKd: 195nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKd: 188nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
Affinity DataKi: 26.4nMAssay Description:Compound was evaluated for its ability to displace [3H]Ins(1,4,5)P3 from membranes prepared from bovine adrenal corticlesMore data for this Ligand-Target Pair
Affinity DataKi: 2.92E+5nMAssay Description:Compound was evaluated for its ability to inhibit Inositol phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Binding affinity against Ins(1,4,5)P3 receptor in swiss 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 598nMAssay Description:Binding affinity towards Inositol 1,4,5-trisphosphate receptor was evaluated by the standard competitive binding assay using 1.25 nM [3H]-D-I(1,4,5)P...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity towards Inositol 1,4,5-trisphosphate receptor was evaluated by the standard competitive binding assay using 1.25 nM [3H]-D-I(1,4,5)P...More data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of Ins(1,3,4,5)P4-PtdIns(3,4,5)P3-specific receptor from Pig cerebellum membraneMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of Ins(1,3,4,5)P4-PtdIns(3,4,5)P3-specific receptor from Pig cerebellum membraneMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of Ins(1,3,4,5)P4-PtdIns(3,4,5)P3-specific receptor from Pig cerebellum membraneMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of Ins(1,3,4,5)P4-PtdIns(3,4,5)P3-specific receptor from Pig cerebellum membraneMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of Ins(1,3,4,5)P4-PtdIns(3,4,5)P3-specific receptor from Pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against Inositol 1,4,5-trisphosphate receptor on bovine adrenal cortex microsomes.More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against Inositol 1,4,5-trisphosphate receptor on bovine adrenal cortex microsomes.More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against Inositol 1,4,5-trisphosphate receptor on bovine adrenal cortex microsomes.More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Binding affinity against Inositol 1,4,5-trisphosphate receptor on bovine adrenal cortex microsomes.More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Inositol 1,4,5-trisphosphate receptor on bovine adrenal cortex microsomes.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Binding affinity against Inositol 1,4,5-trisphosphate receptor on bovine adrenal cortex microsomes.More data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
Affinity DataKd: 3.20E+3nMAssay Description:Dissociation constant of the compound was determined using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 4.60nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 213nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 1.08E+3nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 2.10nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 2.04E+3nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 24.8nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 4.43E+3nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 394nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 11.3nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 49.2nMAssay Description:Agonistic potency at rat IP3 type 1 receptor expressed in chicken DT40 cellsMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 4.90nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataEC50: 42nMAssay Description:Agonist activity at rat recombinant IP3R1 expressed in chicken DT40 cells assessed as calcium release from intracellular storesMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataKd: 12.5nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 1(Rattus norvegicus)
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataKd: 1.26nMAssay Description:Displacement of [3H]IP3 from full-length rat recombinant IP3R1 expressed in chicken DT40 cells by equilibrium competitive binding assayMore data for this Ligand-Target Pair