Compile Data Set for Download or QSAR
maximum 50k data
Found 187 Enz. Inhib. hit(s) with Target = 'Intermediate conductance calcium-activated potassium channel protein 4'
LigandPNGBDBM205004(US9556132, 2 | process for preparing 2-{2-[1-(2-fl...)
Affinity DataIC50:  5.90E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205081(US9556132, 65 | process for preparing 1-phenyl-5-(...)
Affinity DataIC50:  890nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205016(US9556132, 3 | process for preparing 5-[2-(2-ethox...)
Affinity DataIC50:  37nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205019(US9556132, 4 | process for preparing 1-(2-fluoroph...)
Affinity DataIC50:  30nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205022(US9556132, 40 | US9556132, 5)
Affinity DataIC50:  290nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205028(US9556132, 6 | process for preparing 5-{2-[2-(cycl...)
Affinity DataIC50:  710nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205030(US9556132, 7 | process for preparing 2-(2-{2-[1-(2...)
Affinity DataIC50:  16nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205044(US9556132, 8 | process for preparing methyl 2-(2-{...)
Affinity DataIC50:  590nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205045(US9556132, 9 | process for preparing 1-(2-fluoroph...)
Affinity DataIC50:  770nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205049(US9556132, 12 | process for preparing 5-{2-[2-(flu...)
Affinity DataIC50:  300nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205050(US9556132, 13 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  110nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205051(US9556132, 14 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  460nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205052(US9556132, 15 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  1.70E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205053(US9556132, 16 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  190nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205054(US9556132, 17 | process for preparing 2-(2-{2-[1-(...)
Affinity DataIC50:  1.00E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205055(US9556132, 19 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  510nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205056(US9556132, 20 | process for preparing 5-[2-(2-ethy...)
Affinity DataIC50:  290nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205057(US9556132, 21 | process for preparing 2-{2-[1-(2-f...)
Affinity DataIC50:  550nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205058(US9556132, 22 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  1.70E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205059(US9556132, 23 | process for preparing 5-[2-(2-brom...)
Affinity DataIC50:  550nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205060(US9556132, 24 | US9556132, 25 | process for prepar...)
Affinity DataIC50:  360nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205060(US9556132, 24 | US9556132, 25 | process for prepar...)
Affinity DataIC50:  700nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205062(US9556132, 26 | process for preparing 2-{2-[1-(2-f...)
Affinity DataIC50:  820nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205063(US9556132, 27 | process for preparing 2-{2-[1-(2-f...)
Affinity DataIC50:  900nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205064(US9556132, 28 | process for preparing (2-{2-[1-(2-...)
Affinity DataIC50:  770nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205065(US9556132, 29 | process for preparing 1-(2-fluorop...)
Affinity DataIC50:  58nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205066(US9556132, 30 | process for preparing (e)-n-[(2-{2...)
Affinity DataIC50:  57nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205067(US9556132, 31 | process for preparing 2-{2-[1-(2-f...)
Affinity DataIC50:  110nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205068(US9556132, 32 | process for preparing 5-{2-[2-(dif...)
Affinity DataIC50:  870nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205069(US9556132, 33 | process for preparing 5-{2-[2-(flu...)
Affinity DataIC50:  17nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205022(US9556132, 40 | US9556132, 5)
Affinity DataIC50:  800nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205071(US9556132, 42 | process for preparing 2-{2-[1-(2-f...)
Affinity DataIC50:  680nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205072(US9556132, 48 | process for preparing 1-(2-chlorop...)
Affinity DataIC50:  1.00E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205073(US9556132, 49 | process for preparing 1-(2-chlorop...)
Affinity DataIC50:  540nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205074(US9556132, 51 | process for preparing 1-(2-methoxy...)
Affinity DataIC50:  1.20E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205075(US9556132, 53 | process for preparing 2-{5-[2-(2-m...)
Affinity DataIC50:  1.20E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205076(US9556132, 54 | process for preparing 5-[2-(2-fluo...)
Affinity DataIC50:  780nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205077(US9556132, 56 | process for preparing 2-{5-[2-(2-m...)
Affinity DataIC50:  64nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205078(US9556132, 58 | process for preparing 1-[2-(difluo...)
Affinity DataIC50:  1.10E+3nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205079(US9556132, 59 | process for preparing 1-[2-(difluo...)
Affinity DataIC50:  69nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM205080(US9556132, 62 | process for preparing 2-(5-{2-[2-(...)
Affinity DataIC50:  210nMpH: 7.3Assay Description:Human HEK293 cells over-expressing human IK are grown in culture medium (DMEM supplemented with 10% foetal bovine serum), in polystyrene culture flas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50371391(SENICAPOC)
Affinity DataIC50:  6nMAssay Description:Inhibition of Kca 3.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019900(CHEMBL3287205 | US9533999, i-5)
Affinity DataIC50:  49nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019901(CHEMBL3287206 | US9533999, i-34)
Affinity DataIC50:  96nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019902(CHEMBL3287207)
Affinity DataIC50:  39nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019903(CHEMBL3287208 | US9533999, i-40)
Affinity DataIC50:  48nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019904(CHEMBL3287209 | US9533999, ii-1)
Affinity DataIC50:  52nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019905(CHEMBL3287210 | US9533999, ii-4)
Affinity DataIC50:  41nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019906(CHEMBL3287211 | US9533999, ii-11)
Affinity DataIC50:  66nMAssay Description:Inhibition of human KCa3.1 overexpressed in HEK293 cells assessed as thallium influx preincubated for 15 mins followed by thallium/ionomycin addition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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