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Found 482 Enz. Inhib. hit(s) with Target = 'Microtubule-associated protein tau'
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142851(US8940738, 7)
Affinity DataIC50:  78.3nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142850(US8940738, 6)
Affinity DataIC50:  10.1nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142849(US8940738, 5)
Affinity DataIC50:  33.1nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142848(US8940738, 4)
Affinity DataIC50:  8.40nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142847(US8940738, 3)
Affinity DataIC50:  33.4nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142854(US8940738, 10)
Affinity DataIC50:  165nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142852(US8940738, 8)
Affinity DataIC50:  75.3nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142846(US8940738, 2)
Affinity DataIC50:  19.7nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142845(US8940738, 1)
Affinity DataIC50:  15.5nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142855(US8940738, 11)
Affinity DataIC50:  6.70nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Bos taurus (Bovine))
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM142853(US8940738, 9)
Affinity DataIC50:  608nMpH: 6.5 T: 2°CAssay Description:A mixture containing 100 mM MES-sodium hydroxide (pH 6.5), 1 mM magnesium acetate, 0.5 mM EGTA, 5 mM beta-mercaptoethanol, 0.02% Tween 20, 10% glycer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281656(US10022461, Compound 126)
Affinity DataKi:  0.180nM ΔG°:  -55.6kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281558(US10022461, Compound 9)
Affinity DataKi:  0.220nM ΔG°:  -55.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281645(US10022461, Compound 115)
Affinity DataKi:  0.224nM ΔG°:  -55.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281560(US10022461, Compound 12)
Affinity DataKi:  0.290nM ΔG°:  -54.4kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281561(US10022461, Compound 13)
Affinity DataKi:  0.290nM ΔG°:  -54.4kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281633(US10022461, Compound 103)
Affinity DataKi:  0.320nM ΔG°:  -54.2kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281563(US10022461, Compound 14-1)
Affinity DataKi:  0.330nM ΔG°:  -54.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281609(US10022461, Compound 59)
Affinity DataKi:  0.330nM ΔG°:  -54.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281635(US10022461, Compound 105)
Affinity DataKi:  0.383nM ΔG°:  -53.7kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281559(US10022461, Compound 11-5)
Affinity DataKi:  0.400nM ΔG°:  -53.6kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281565(US10022461, Compound 16)
Affinity DataKi:  0.410nM ΔG°:  -53.6kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281639(US10022461, Compound 109)
Affinity DataKi:  0.423nM ΔG°:  -53.5kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281567(US10022461, Compound 18)
Affinity DataKi:  0.430nM ΔG°:  -53.5kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281566(US10022461, Compound 17)
Affinity DataKi:  0.430nM ΔG°:  -53.5kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281649(US10022461, Compound 119)
Affinity DataKi:  0.438nM ΔG°:  -53.4kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281557(US10022461, Compound 8)
Affinity DataKi:  0.480nM ΔG°:  -53.2kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281623(US10022461, Compound 75)
Affinity DataKi:  0.480nM ΔG°:  -53.2kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281644(US10022461, Compound 114)
Affinity DataKi:  0.494nM ΔG°:  -53.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281651(US10022461, Compound 121)
Affinity DataKi:  0.512nM ΔG°:  -53.0kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281626(US10022461, Compound 93)
Affinity DataKi:  0.530nM ΔG°:  -52.9kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281564(US10022461, Compound 15)
Affinity DataKi:  0.530nM ΔG°:  -52.9kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281555(US10022461, Compound 6)
Affinity DataKi:  0.540nM ΔG°:  -52.9kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281630(US10022461, Compound 99)
Affinity DataKi:  0.550nM ΔG°:  -52.9kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281568(US10022461, Compound 19)
Affinity DataKi:  0.620nM ΔG°:  -52.6kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281599(US10022461, Compound 49)
Affinity DataKi:  0.670nM ΔG°:  -52.4kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281642(US10022461, Compound 112)
Affinity DataKi:  0.672nM ΔG°:  -52.4kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281638(US10022461, Compound 108)
Affinity DataKi:  0.677nM ΔG°:  -52.3kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281624(US10022461, Compound 88)
Affinity DataKi:  0.690nM ΔG°:  -52.3kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281569(US10022461, Compound 20)
Affinity DataKi:  0.75nM ΔG°:  -52.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281600(US10022461, Compound 50)
Affinity DataKi:  0.75nM ΔG°:  -52.1kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281622(US10022461, Compound 72)
Affinity DataKi:  0.760nM ΔG°:  -52.0kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281643(US10022461, Compound 113)
Affinity DataKi:  0.784nM ΔG°:  -52.0kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281601(US10022461, Compound 51)
Affinity DataKi:  0.870nM ΔG°:  -51.7kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281628(US10022461, Compound 95)
Affinity DataKi:  0.960nM ΔG°:  -51.5kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281602(US10022461, Compound 52)
Affinity DataKi:  0.980nM ΔG°:  -51.4kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281603(US10022461, Compound 53)
Affinity DataKi:  1.02nM ΔG°:  -51.3kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281604(US10022461, Compound 54)
Affinity DataKi:  1.05nM ΔG°:  -51.2kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281631(US10022461, Compound 100)
Affinity DataKi:  1.06nM ΔG°:  -51.2kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM281654(US10022461, Compound 124)
Affinity DataKi:  1.07nM ΔG°:  -51.2kJ/molepH: 7.4 T: 2°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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