Compile Data Set for Download or QSAR
maximum 50k data
Found 269 Enz. Inhib. hit(s) with Target = 'Peregrin'
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148549(4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-ox...)
Affinity DataIC50:  270nMpH: 7.4 T: 2°CAssay Description:Assays were performed as described previously with minor modifications(Philpott et al., 2011). All reagents were diluted in 25 mM HEPES, 100 mM NaCl,...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032927(CHEMBL3356143 | N-[2,3-Dihydro-1,3-dimethyl-2-oxo-...)
Affinity DataIC50:  172nMpH: 7.4 T: 2°CAssay Description:Assays were performed as described previously with minor modifications(Philpott et al., 2011). All reagents were diluted in 25 mM HEPES, 100 mM NaCl,...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50157570(4-cyano-N-(1,3-dimethyl-2-oxoquinolin-6-yl)-2-meth...)
Affinity DataIC50:  114nMpH: 7.4 T: 2°CAssay Description:Assays were performed as described previously with minor modifications(Philpott et al., 2011). All reagents were diluted in 25 mM HEPES, 100 mM NaCl,...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540508(CHEMBL4648548)
Affinity DataKi:  251nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50098311(CHEMBL3590408)
Affinity DataKi:  5.01E+3nMAssay Description:Binding affinity to BRPF1 (unknown origin) by BROMOscan panel based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50572130(CHEMBL4864027)
Affinity DataKi:  5.01E+3nMAssay Description:Inhibition of human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540519(CHEMBL4635895)
Affinity DataKi:  6.31E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540521(CHEMBL4632508)
Affinity DataKi:  7.94E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540520(CHEMBL4644517)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540518(CHEMBL4646338)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540517(CHEMBL4642556)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540516(CHEMBL4635826)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540514(CHEMBL4636297)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540513(CHEMBL4645418)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540512(CHEMBL4642886)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540515(CHEMBL4635892)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540523(CHEMBL4634319)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50540522(CHEMBL4639574)
Affinity DataKi: <3.16E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50028142(CHEMBL2177300)
Affinity DataIC50: <4nMAssay Description:Inhibition of human BRPF1 by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032909(CHEMBL1361770)
Affinity DataIC50:  631nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032910(CHEMBL3356147)
Affinity DataIC50:  3.16E+3nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032911(CHEMBL1535485)
Affinity DataIC50:  3.16E+3nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032912(CHEMBL1522313)
Affinity DataIC50:  980nMAssay Description:Binding affinity to NanoLuc-tagged BRPF1 isoform 1 bromodomain (625-735 aa) (unknown origin) expressed in HEK293 cells co-transfected with histone H3...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032912(CHEMBL1522313)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity to NanoLuc-tagged BRPF1 isoform 1 bromodomain (625-735 aa) (unknown origin) expressed in HEK293 cells co-transfected with histone H3...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032913(CHEMBL1487662)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032921(CHEMBL1444120)
Affinity DataIC50:  200nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032912(CHEMBL1522313)
Affinity DataIC50:  79nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032920(CHEMBL3356138)
Affinity DataIC50:  631nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032919(CHEMBL3356139)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032918(CHEMBL3356140)
Affinity DataIC50:  100nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032917(CHEMBL1724375)
Affinity DataIC50:  100nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032916(CHEMBL1357836)
Affinity DataIC50:  316nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032915(CHEMBL3356141)
Affinity DataIC50:  631nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032914(CHEMBL3356142)
Affinity DataIC50:  398nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032927(CHEMBL3356143 | N-[2,3-Dihydro-1,3-dimethyl-2-oxo-...)
Affinity DataIC50:  50nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032922(CHEMBL1701516)
Affinity DataIC50:  316nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032923(CHEMBL3356144)
Affinity DataIC50:  794nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032924(CHEMBL1396002)
Affinity DataIC50:  126nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032928(CHEMBL3356145)
Affinity DataIC50:  126nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032925(CHEMBL3356146)
Affinity DataIC50:  1.59E+3nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50032926(CHEMBL1702128)
Affinity DataIC50:  2.51E+3nMAssay Description:Binding affinity to 6H-Flag-tagged Tev-BRPF1 (622-738 aa) (unknown origin) by TR-FRET competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50098250(CHEMBL3590389)
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to BRPF1 in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50098305(CHEMBL3590405)
Affinity DataKd:  2.51E+4nMAssay Description:Binding affinity to BRPF1 in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50098311(CHEMBL3590408)
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to BRPF1 in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148460(CHEMBL1346130)
Affinity DataIC50:  330nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148461(CHEMBL3770652)
Affinity DataIC50:  590nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148462(CHEMBL3770886)
Affinity DataIC50:  420nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148463(CHEMBL3770971)
Affinity DataIC50:  270nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148464(CHEMBL3771106)
Affinity DataIC50:  310nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
Oxford University

LigandPNGBDBM50148465(CHEMBL3771151)
Affinity DataIC50:  290nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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