Compile Data Set for Download or QSAR
maximum 50k data
Found 1872 Enz. Inhib. hit(s) with Target = 'Urokinase-type plasminogen activator'
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92292(uPa_17)
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14142(2-{5-[amino(iminiumyl)methyl]-1H-indol-2-yl}-6-phe...)
Affinity DataKi:  8nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14152(6-CHLORO-2-(2-HYDROXY-BIPHENYL-3-YL)-1H-INDOLE-5-C...)
Affinity DataKi:  9nM ΔG°:  -45.5kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92321(uPa_43)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14149(6-fluoro-2-(2-hydroxy-3-{[(1S,2S)-2-methylcyclohex...)
Affinity DataKi:  11nM ΔG°:  -45.0kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92302(uPa_26)
Affinity DataKi:  16nM ΔG°:  -44.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92313(uPa_36)
Affinity DataKi:  18nM ΔG°:  -44.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14150(APC-11417 | CA-12 | CRA-11417 | {amino[6-fluoro-2-...)
Affinity DataKi:  20nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92316(uPa_39)
Affinity DataKi:  21nM ΔG°:  -43.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92304(uPa_28)
Affinity DataKi:  33nM ΔG°:  -42.7kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92287(uPa_10)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92319(uPa_41)
Affinity DataKi:  42nM ΔG°:  -42.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92293(uPa_18)
Affinity DataKi:  59nM ΔG°:  -41.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92308(uPa_31)
Affinity DataKi:  66nM ΔG°:  -41.0kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14156(3-bromo-N-(4-carbamimidoylphenyl)-2-hydroxy-5-meth...)
Affinity DataKi:  77nM ΔG°:  -40.2kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92320(uPa_42)
Affinity DataKi:  94nM ΔG°:  -40.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14148(2-{5-[amino(iminiumyl)methyl]-6-fluoro-1H-1,3-benz...)
Affinity DataKi:  110nM ΔG°:  -39.3kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14146(APC-9008 | {amino[2-(3,5-dichloro-2-hydroxyphenyl)...)
Affinity DataKi:  200nM ΔG°:  -37.9kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14169(4-Iodobenzo[b]thiophene-2-carboxamidine | APC-6860...)
Affinity DataKi:  210nM ΔG°:  -37.7kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14144(2-{5-[amino(iminiumyl)methyl]-1H-1,3-benzodiazol-2...)
Affinity DataKi:  220nM ΔG°:  -37.6kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92318(uPa_40)
Affinity DataKi:  223nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14158(APC-11922 | CHEMBL293260 | N-(4-carbamimidoyl-3-fl...)
Affinity DataKi:  270nM ΔG°:  -37.1kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92305(uPa_29)
Affinity DataKi:  290nM ΔG°:  -37.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14151(APC-9850 | {amino[6-chloro-2-(3,5-dichloro-2-hydro...)
Affinity DataKi:  310nM ΔG°:  -36.8kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14157(APC-10605 | CHEMBL64097 | N-(4-carbamimidoylphenyl...)
Affinity DataKi:  330nM ΔG°:  -36.6kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92294(uPa_19)
Affinity DataKi:  406nM ΔG°:  -36.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14143(2-(2-HYDROXY-BIPHENYL)-1H-BENZOIMIDAZOLE-5-CARBOXA...)
Affinity DataKi:  450nM ΔG°:  -35.9kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50147092(8-Amino-naphthalene-2-carboxamidine | 8-amino-2-na...)
Affinity DataKi:  450nM ΔG°:  -36.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14145(2-{5-[amino(iminiumyl)methyl]-1H-1,3-benzodiazol-2...)
Affinity DataKi:  500nM ΔG°:  -35.6kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14147(APC-10818 | {amino[6-fluoro-2-(2-hydroxy-3-phenylp...)
Affinity DataKi:  590nM ΔG°:  -35.2kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92325(uPa_8)
Affinity DataKi:  610nM ΔG°:  -35.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92289(uPa_12)
Affinity DataKi:  610nM ΔG°:  -35.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  628nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50147085(7-METHOXY-8-[1-(METHYLSULFONYL)-1H-PYRAZOL-4-YL]NA...)
Affinity DataKi:  630nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92317(uPa_4)
Affinity DataKi:  637nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92301(uPa_25)
Affinity DataKi:  665nM ΔG°:  -35.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92296(uPa_20)
Affinity DataKi:  769nM ΔG°:  -34.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92315(uPa_38)
Affinity DataKi:  777nM ΔG°:  -34.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92322(uPa_44)
Affinity DataKi:  1.25E+3nM ΔG°:  -33.7kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92314(uPa_37)
Affinity DataKi:  1.49E+3nM ΔG°:  -33.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14154(2-{5-[amino(iminiumyl)methyl]-6-chloro-1H-1,3-benz...)
Affinity DataKi:  1.80E+3nM ΔG°:  -32.5kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14153(2-{5-[amino(iminiumyl)methyl]-6-chloro-1H-1,3-benz...)
Affinity DataKi:  2.10E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14170(APC-7377 | Benzo[b]thiophene-2-carboxamidine | [am...)
Affinity DataKi:  2.30E+3nM ΔG°:  -31.9kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92309(uPa_32)
Affinity DataKi:  3.08E+3nM ΔG°:  -31.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92298(uPa_22)
Affinity DataKi:  3.57E+3nM ΔG°:  -31.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  3.80E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92288(uPa_11)
Affinity DataKi:  4.50E+3nM ΔG°:  -30.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138663(2-naphthimidamide | CHEMBL105171 | Naphthalene-2-c...)
Affinity DataKi:  5.91E+3nM ΔG°:  -29.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM14159(APC-11421 | CHEMBL62897 | N-(4-carbamimidoyl-3-chl...)
Affinity DataKi:  6.00E+3nM ΔG°:  -29.5kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
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