Affinity DataKi: 87nM ΔG°: -39.9kJ/molepH: 7.8 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of activated protein kinase C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of activated Protein C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of activated Protein C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of human activated protein C using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of human activated protein C using H-D-Lys(Cbz)-Pro-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of activated protein C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of activated protein C (unknown origin) at 37 degC by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity to human activated protein C assessed as release of p-nitroaniline after 10 to 120 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: >130nMAssay Description:Inhibition of human activated protein kinase C using H-D-Lys(Cbo)-Pro-Arg-pNA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Inhibition of activated protein C (unknown origin) at 37 degC by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Inhibition of activated protein C (unknown origin) at 37 degC by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of human activated protein C using pyroGlu-Pro-Arg-pNA as substrate assessed as release of pNA after 10 to 120 mins by spectrophotometric ...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of activated protein C (unknown origin) at 37 degC by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 223nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Inhibition of activated protein C (unknown origin) at 37 degC by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Inhibition of human activated protein C using H-D-Lys(Cbz)-Pro-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 555nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 564nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 725nMAssay Description:Inhibition of activated protein C (unknown origin) at 37 degC by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 830nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Inhibition of human aPC was determined by the method described in [0092]-[0098] using human activated protein C from Enzyme Research Laboratories at ...More data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Inhibition of human activated protein C using H-D-Lys(Cbz)-Pro-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair