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Compile Data Set for Download or QSAR

Found 430 hits Enz. Inhib. hit(s) with Target = 'Voltage-gated potassium channel subunit Kv7.2'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50529214
PNG
(CHEMBL343822)
Show SMILES Fc1cc(CC2(Cc3ccnc(F)c3)c3ccccc3C(=O)c3ccccc23)ccn1
Show InChI InChI=1S/C26H18F2N2O/c27-23-13-17(9-11-29-23)15-26(16-18-10-12-30-24(28)14-18)21-7-3-1-5-19(21)25(31)20-6-2-4-8-22(20)26/h1-14H,15-16H2
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n/an/a 48n/an/an/an/an/an/a



Marquette University

Curated by ChEMBL


Assay Description
Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assay


Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126681
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50529215
PNG
(CHEBI:35046 | CHEMBL342375)
Show SMILES O=C1c2ccccc2C(Cc2ccncc2)(Cc2ccncc2)c2ccccc12
Show InChI InChI=1S/C26H20N2O/c29-25-21-5-1-3-7-23(21)26(17-19-9-13-27-14-10-19,18-20-11-15-28-16-12-20)24-8-4-2-6-22(24)25/h1-16H,17-18H2
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n/an/a 55n/an/an/an/an/an/a



Marquette University

Curated by ChEMBL


Assay Description
Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assay


Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126681
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84190
PNG
((2,6-dimethyl-4-morpholinyl)-(6-methyl-2-phenyl-4-...)
Show SMILES CC1CN(CC(C)O1)C(=O)c1cc(nc2ccc(C)cc12)-c1ccccc1
Show InChI InChI=1S/C23H24N2O2/c1-15-9-10-21-19(11-15)20(12-22(24-21)18-7-5-4-6-8-18)23(26)25-13-16(2)27-17(3)14-25/h4-12,16-17H,13-14H2,1-3H3
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n/an/a 68.1n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84168
PNG
(2-[2,4-bis(chloranyl)phenoxy]-N-cyclohexyl-N-pyrid...)
Show SMILES Clc1ccc(OCC(=O)N(C2CCCCC2)c2ccccn2)c(Cl)c1
Show InChI InChI=1S/C19H20Cl2N2O2/c20-14-9-10-17(16(21)12-14)25-13-19(24)23(15-6-2-1-3-7-15)18-8-4-5-11-22-18/h4-5,8-12,15H,1-3,6-7,13H2
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n/an/a 69.9n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395464
PNG
(CHEMBL2164048)
Show SMILES CC[C@H](C(=O)Nc1ccccc1N1CCCC1)c1ccccc1
Show InChI InChI=1S/C20H24N2O/c1-2-17(16-10-4-3-5-11-16)20(23)21-18-12-6-7-13-19(18)22-14-8-9-15-22/h3-7,10-13,17H,2,8-9,14-15H2,1H3,(H,21,23)/t17-/m0/s1
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n/an/a 70n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84176
PNG
(2-[benzenesulfonyl(methyl)amino]-N-(2-methylphenyl...)
Show SMILES CN(c1ccccc1C(=O)Nc1ccccc1C)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C21H20N2O3S/c1-16-10-6-8-14-19(16)22-21(24)18-13-7-9-15-20(18)23(2)27(25,26)17-11-4-3-5-12-17/h3-15H,1-2H3,(H,22,24)
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n/an/a 92.3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84171
PNG
(MLS000516664 | N-(2-morpholin-4-ylphenyl)-2-(3,4,5...)
Show SMILES COc1cc(cc(OC)c1OC)-c1cc(C(=O)Nc2ccccc2N2CCOCC2)c2ccccc2n1
Show InChI InChI=1S/C29H29N3O5/c1-34-26-16-19(17-27(35-2)28(26)36-3)24-18-21(20-8-4-5-9-22(20)30-24)29(33)31-23-10-6-7-11-25(23)32-12-14-37-15-13-32/h4-11,16-18H,12-15H2,1-3H3,(H,31,33)
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n/an/a 110n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2/Kv7.3


(Homo sapiens (Human))
BDBM50395464
PNG
(CHEMBL2164048)
Show SMILES CC[C@H](C(=O)Nc1ccccc1N1CCCC1)c1ccccc1
Show InChI InChI=1S/C20H24N2O/c1-2-17(16-10-4-3-5-11-16)20(23)21-18-12-6-7-13-19(18)22-14-8-9-15-22/h3-7,10-13,17H,2,8-9,14-15H2,1H3,(H,21,23)/t17-/m0/s1
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n/an/a 120n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2/Q3 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395501
PNG
(CHEMBL2163658)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(OC)c1
Show InChI InChI=1S/C21H26N2O2/c1-3-18(16-9-8-10-17(15-16)25-2)21(24)22-19-11-4-5-12-20(19)23-13-6-7-14-23/h4-5,8-12,15,18H,3,6-7,13-14H2,1-2H3,(H,22,24)
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n/an/a 120n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395505
PNG
(CHEMBL2164068)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(F)cc1
Show InChI InChI=1S/C20H23FN2O/c1-2-17(15-9-11-16(21)12-10-15)20(24)22-18-7-3-4-8-19(18)23-13-5-6-14-23/h3-4,7-12,17H,2,5-6,13-14H2,1H3,(H,22,24)
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n/an/a 130n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50529213
PNG
(CHEMBL4465132)
Show SMILES Fc1cncc(F)c1CC1(Cc2ccnnc2)c2ccccc2C(=O)c2ccccc12
Show InChI InChI=1S/C25H17F2N3O/c26-22-14-28-15-23(27)19(22)12-25(11-16-9-10-29-30-13-16)20-7-3-1-5-17(20)24(31)18-6-2-4-8-21(18)25/h1-10,13-15H,11-12H2
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n/an/a 160n/an/an/an/an/an/a



Marquette University

Curated by ChEMBL


Assay Description
Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assay


Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126681
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84184
PNG
(2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide | 2...)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1
Show InChI InChI=1S/C20H24N2O/c1-2-17(16-10-4-3-5-11-16)20(23)21-18-12-6-7-13-19(18)22-14-8-9-15-22/h3-7,10-13,17H,2,8-9,14-15H2,1H3,(H,21,23)
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n/an/a 161n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM84184
PNG
(2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide | 2...)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1
Show InChI InChI=1S/C20H24N2O/c1-2-17(16-10-4-3-5-11-16)20(23)21-18-12-6-7-13-19(18)22-14-8-9-15-22/h3-7,10-13,17H,2,8-9,14-15H2,1H3,(H,21,23)
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n/an/a 163n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395508
PNG
(CHEMBL2164062)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(F)c(F)c1
Show InChI InChI=1S/C20H22F2N2O/c1-2-15(14-9-10-16(21)17(22)13-14)20(25)23-18-7-3-4-8-19(18)24-11-5-6-12-24/h3-4,7-10,13,15H,2,5-6,11-12H2,1H3,(H,23,25)
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n/an/a 170n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50529212
PNG
(CHEMBL4471453)
Show SMILES Fc1cncc(F)c1CC1(Cc2c(F)cncc2F)c2ccccc2C(=O)c2ccccc12
Show InChI InChI=1S/C26H16F4N2O/c27-21-11-31-12-22(28)17(21)9-26(10-18-23(29)13-32-14-24(18)30)19-7-3-1-5-15(19)25(33)16-6-2-4-8-20(16)26/h1-8,11-14H,9-10H2
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n/an/a 200n/an/an/an/an/an/a



Marquette University

Curated by ChEMBL


Assay Description
Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assay


Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126681
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395481
PNG
(CHEMBL2163667)
Show SMILES CCC(C(=O)Nc1ccc(cc1)N1CCCC1)c1ccccc1
Show InChI InChI=1S/C20H24N2O/c1-2-19(16-8-4-3-5-9-16)20(23)21-17-10-12-18(13-11-17)22-14-6-7-15-22/h3-5,8-13,19H,2,6-7,14-15H2,1H3,(H,21,23)
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n/an/a 210n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84160
PNG
(4-methyl-N-[3-methyl-1-(o-anisylcarbamoyl)butyl]cy...)
Show SMILES COc1ccccc1CNC(=O)C(CC(C)C)NC(=O)C1CCC(C)CC1
Show InChI InChI=1S/C22H34N2O3/c1-15(2)13-19(24-21(25)17-11-9-16(3)10-12-17)22(26)23-14-18-7-5-6-8-20(18)27-4/h5-8,15-17,19H,9-14H2,1-4H3,(H,23,26)(H,24,25)
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n/an/a 210n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395500
PNG
(CHEMBL2163659)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(Cl)c1
Show InChI InChI=1S/C20H23ClN2O/c1-2-17(15-8-7-9-16(21)14-15)20(24)22-18-10-3-4-11-19(18)23-12-5-6-13-23/h3-4,7-11,14,17H,2,5-6,12-13H2,1H3,(H,22,24)
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n/an/a 240n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84164
PNG
(2-Ethyl-3,6-dimethyl-quinoline-4-carboxylic acid (...)
Show SMILES CCc1nc2ccc(C)cc2c(C(=O)NC2CCCCC2C)c1C
Show InChI InChI=1S/C21H28N2O/c1-5-17-15(4)20(16-12-13(2)10-11-19(16)22-17)21(24)23-18-9-7-6-8-14(18)3/h10-12,14,18H,5-9H2,1-4H3,(H,23,24)
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n/an/a 254n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395518
PNG
(CHEMBL2164049)
Show SMILES CC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1
Show InChI InChI=1S/C19H22N2O/c1-15(16-9-3-2-4-10-16)19(22)20-17-11-5-6-12-18(17)21-13-7-8-14-21/h2-6,9-12,15H,7-8,13-14H2,1H3,(H,20,22)
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n/an/a 260n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395498
PNG
(CHEMBL2163662)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(Cl)cc1
Show InChI InChI=1S/C20H23ClN2O/c1-2-17(15-9-11-16(21)12-10-15)20(24)22-18-7-3-4-8-19(18)23-13-5-6-14-23/h3-4,7-12,17H,2,5-6,13-14H2,1H3,(H,22,24)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395515
PNG
(CHEMBL2164054)
Show SMILES CCCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1
Show InChI InChI=1S/C21H26N2O/c1-2-10-18(17-11-4-3-5-12-17)21(24)22-19-13-6-7-14-20(19)23-15-8-9-16-23/h3-7,11-14,18H,2,8-10,15-16H2,1H3,(H,22,24)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395506
PNG
(CHEMBL2164066)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(C)c1
Show InChI InChI=1S/C21H26N2O/c1-3-18(17-10-8-9-16(2)15-17)21(24)22-19-11-4-5-12-20(19)23-13-6-7-14-23/h4-5,8-12,15,18H,3,6-7,13-14H2,1-2H3,(H,22,24)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395514
PNG
(CHEMBL2164055)
Show SMILES O=C(Nc1ccccc1N1CCCC1)C1CCc2ccccc12
Show InChI InChI=1S/C20H22N2O/c23-20(17-12-11-15-7-1-2-8-16(15)17)21-18-9-3-4-10-19(18)22-13-5-6-14-22/h1-4,7-10,17H,5-6,11-14H2,(H,21,23)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395507
PNG
(CHEMBL2164064)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(F)c1
Show InChI InChI=1S/C20H23FN2O/c1-2-17(15-8-7-9-16(21)14-15)20(24)22-18-10-3-4-11-19(18)23-12-5-6-13-23/h3-4,7-11,14,17H,2,5-6,12-13H2,1H3,(H,22,24)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395499
PNG
(CHEMBL2163661)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(OC)cc1
Show InChI InChI=1S/C21H26N2O2/c1-3-18(16-10-12-17(25-2)13-11-16)21(24)22-19-8-4-5-9-20(19)23-14-6-7-15-23/h4-5,8-13,18H,3,6-7,14-15H2,1-2H3,(H,22,24)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395502
PNG
(CHEMBL2163657)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(c1)C(F)(F)F
Show InChI InChI=1S/C21H23F3N2O/c1-2-17(15-8-7-9-16(14-15)21(22,23)24)20(27)25-18-10-3-4-11-19(18)26-12-5-6-13-26/h3-4,7-11,14,17H,2,5-6,12-13H2,1H3,(H,25,27)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395497
PNG
(CHEMBL2163664)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1F
Show InChI InChI=1S/C20H23FN2O/c1-2-15(16-9-3-4-10-17(16)21)20(24)22-18-11-5-6-12-19(18)23-13-7-8-14-23/h3-6,9-12,15H,2,7-8,13-14H2,1H3,(H,22,24)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50395504
PNG
(CHEMBL2164069)
Show SMILES CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C20H22Cl2N2O/c1-2-15(14-9-10-16(21)17(22)13-14)20(25)23-18-7-3-4-8-19(18)24-11-5-6-12-24/h3-4,7-10,13,15H,2,5-6,11-12H2,1H3,(H,23,25)
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Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84157
PNG
(4-[(3,4-dimethylphenyl)carbamoyl-(2-methoxyethyl)a...)
Show SMILES CCOC(=O)N1CCC(CC1)N(CCOC)C(=O)Nc1ccc(C)c(C)c1
Show InChI InChI=1S/C20H31N3O4/c1-5-27-20(25)22-10-8-18(9-11-22)23(12-13-26-4)19(24)21-17-7-6-15(2)16(3)14-17/h6-7,14,18H,5,8-13H2,1-4H3,(H,21,24)
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84185
PNG
(MLS001157683 | N-[2-(3,4-dimethoxyphenyl)ethyl]-N,...)
Show SMILES COc1ccc(CCN(C)C(=O)c2cc(nc3ccc(C)cc23)-c2ccccc2)cc1OC
Show InChI InChI=1S/C28H28N2O3/c1-19-10-12-24-22(16-19)23(18-25(29-24)21-8-6-5-7-9-21)28(31)30(2)15-14-20-11-13-26(32-3)27(17-20)33-4/h5-13,16-18H,14-15H2,1-4H3
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n/an/a 478n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84159
PNG
(MLS000520753 | N-(4-oxidanylidene-2-phenacylsulfan...)
Show SMILES O=C(CSc1nc2ccccc2c(=O)n1NC(=O)c1ccccc1)c1ccccc1
Show InChI InChI=1S/C23H17N3O3S/c27-20(16-9-3-1-4-10-16)15-30-23-24-19-14-8-7-13-18(19)22(29)26(23)25-21(28)17-11-5-2-6-12-17/h1-14H,15H2,(H,25,28)
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM50529217
PNG
(CHEMBL4447214)
Show SMILES Cc1cc(CC2(Cc3ccnc(C)c3)c3ccccc3C(=O)c3ccccc23)ccn1
Show InChI InChI=1S/C28H24N2O/c1-19-15-21(11-13-29-19)17-28(18-22-12-14-30-20(2)16-22)25-9-5-3-7-23(25)27(31)24-8-4-6-10-26(24)28/h3-16H,17-18H2,1-2H3
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Marquette University

Curated by ChEMBL


Assay Description
Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assay


Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126681
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84186
PNG
(MLS001157673 | N-[2-(3,4-dimethoxyphenyl)ethyl]-N-...)
Show SMILES COc1ccc(CCN(C)C(=O)c2cc(nc3ccccc23)-c2ccc(C)cc2)cc1OC
Show InChI InChI=1S/C28H28N2O3/c1-19-9-12-21(13-10-19)25-18-23(22-7-5-6-8-24(22)29-25)28(31)30(2)16-15-20-11-14-26(32-3)27(17-20)33-4/h5-14,17-18H,15-16H2,1-4H3
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84188
PNG
((2,6-dimethyl-4-morpholinyl)-[2-(5-methyl-2-furany...)
Show SMILES CC1CN(CC(C)O1)C(=O)c1cc(nc2ccccc12)-c1ccc(C)o1
Show InChI InChI=1S/C21H22N2O3/c1-13-8-9-20(26-13)19-10-17(16-6-4-5-7-18(16)22-19)21(24)23-11-14(2)25-15(3)12-23/h4-10,14-15H,11-12H2,1-3H3
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84180
PNG
((2,6-dimethyl-4-quinolinyl)-[3-[4-(2-methylphenyl)...)
Show SMILES Cc1ccc2nc(C)cc(C(=O)N3CCCC(C3)N3CCN(CC3)c3ccccc3C)c2c1
Show InChI InChI=1S/C28H34N4O/c1-20-10-11-26-24(17-20)25(18-22(3)29-26)28(33)32-12-6-8-23(19-32)30-13-15-31(16-14-30)27-9-5-4-7-21(27)2/h4-5,7,9-11,17-18,23H,6,8,12-16,19H2,1-3H3
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM51335
PNG
(2-bromanyl-N-(2,3-dimethylphenyl)-3,4,5-trimethoxy...)
Show SMILES COc1cc(C(=O)Nc2cccc(C)c2C)c(Br)c(OC)c1OC
Show InChI InChI=1S/C18H20BrNO4/c1-10-7-6-8-13(11(10)2)20-18(21)12-9-14(22-3)16(23-4)17(24-5)15(12)19/h6-9H,1-5H3,(H,20,21)
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84177
PNG
(MLS001171558 | N-benzyl-N-methyl-2-(3,4,5-trimetho...)
Show SMILES COc1cc(cc(OC)c1OC)-c1cc(C(=O)N(C)Cc2ccccc2)c2ccccc2n1
Show InChI InChI=1S/C27H26N2O4/c1-29(17-18-10-6-5-7-11-18)27(30)21-16-23(28-22-13-9-8-12-20(21)22)19-14-24(31-2)26(33-4)25(15-19)32-3/h5-16H,17H2,1-4H3
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84165
PNG
(2-Ethyl-6-fluoro-3-methyl-quinoline-4-carboxylic a...)
Show SMILES CCc1nc2ccc(F)cc2c(C(=O)NC2CCCCC2C)c1C
Show InChI InChI=1S/C20H25FN2O/c1-4-16-13(3)19(15-11-14(21)9-10-18(15)22-16)20(24)23-17-8-6-5-7-12(17)2/h9-12,17H,4-8H2,1-3H3,(H,23,24)
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84189
PNG
(2-(2-chloranyl-4-fluoranyl-phenoxy)-N-(2-piperidin...)
Show SMILES Fc1ccc(OCC(=O)Nc2ccccc2C(=O)N2CCCCC2)c(Cl)c1
Show InChI InChI=1S/C20H20ClFN2O3/c21-16-12-14(22)8-9-18(16)27-13-19(25)23-17-7-3-2-6-15(17)20(26)24-10-4-1-5-11-24/h2-3,6-9,12H,1,4-5,10-11,13H2,(H,23,25)
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84175
PNG
(MLS000757674 | N-[[5-(diethylsulfamoyl)-2-(4-morph...)
Show SMILES CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=S)NC(=O)c2ccco2)c1
Show InChI InChI=1S/C20H26N4O5S2/c1-3-24(4-2)31(26,27)15-7-8-17(23-9-12-28-13-10-23)16(14-15)21-20(30)22-19(25)18-6-5-11-29-18/h5-8,11,14H,3-4,9-10,12-13H2,1-2H3,(H2,21,22,25,30)
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Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM77244
PNG
(2-[[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]m...)
Show SMILES COc1cccc(c1)-c1nc(CS(=O)(=O)CC(=O)NC2CCCc3ccccc23)c(C)o1
Show InChI InChI=1S/C24H26N2O5S/c1-16-22(26-24(31-16)18-9-5-10-19(13-18)30-2)14-32(28,29)15-23(27)25-21-12-6-8-17-7-3-4-11-20(17)21/h3-5,7,9-11,13,21H,6,8,12,14-15H2,1-2H3,(H,25,27)
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n/an/a 869n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM61006
PNG
(4-[(3,4-dichlorophenyl)carbamoyl-(2-methoxyethyl)a...)
Show SMILES CCOC(=O)N1CCC(CC1)N(CCOC)C(=O)Nc1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C18H25Cl2N3O4/c1-3-27-18(25)22-8-6-14(7-9-22)23(10-11-26-2)17(24)21-13-4-5-15(19)16(20)12-13/h4-5,12,14H,3,6-11H2,1-2H3,(H,21,24)
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n/an/a 990n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84150
PNG
(2-(2-methyl-3-oxidanylidene-1,4-benzoxazin-4-yl)-N...)
Show SMILES CC1Oc2ccccc2N(CC(=O)N(Cc2ccccc2)Cc2ccccn2)C1=O
Show InChI InChI=1S/C24H23N3O3/c1-18-24(29)27(21-12-5-6-13-22(21)30-18)17-23(28)26(15-19-9-3-2-4-10-19)16-20-11-7-8-14-25-20/h2-14,18H,15-17H2,1H3
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n/an/a 1.00E+3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84158
PNG
(3-(4-ethylphenyl)-1-(2-furanylmethyl)-1-(1-thiophe...)
Show SMILES CCc1ccc(NC(=O)N(Cc2ccco2)C(C)c2cccs2)cc1
Show InChI InChI=1S/C20H22N2O2S/c1-3-16-8-10-17(11-9-16)21-20(23)22(14-18-6-4-12-24-18)15(2)19-7-5-13-25-19/h4-13,15H,3,14H2,1-2H3,(H,21,23)
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n/an/a 1.04E+3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84161
PNG
(1-tert-Butyl-4-[1-(4-chloro-benzyl)-1H-benzoimidaz...)
Show SMILES CC(C)(C)N1CC(CC1=O)c1nc2ccccc2n1Cc1ccc(Cl)cc1
Show InChI InChI=1S/C22H24ClN3O/c1-22(2,3)26-14-16(12-20(26)27)21-24-18-6-4-5-7-19(18)25(21)13-15-8-10-17(23)11-9-15/h4-11,16H,12-14H2,1-3H3
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n/an/a 1.23E+3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
KCNQ (Kv7) potassium channel


(Homo sapiens (Human))
BDBM84166
PNG
(2-phenyl-N-(2-phenylphenyl)butanamide | 2-phenyl-N...)
Show SMILES CCC(C(=O)Nc1ccccc1-c1ccccc1)c1ccccc1
Show InChI InChI=1S/C22H21NO/c1-2-19(17-11-5-3-6-12-17)22(24)23-21-16-10-9-15-20(21)18-13-7-4-8-14-18/h3-16,19H,2H2,1H3,(H,23,24)
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antibodypedia
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n/an/a 1.32E+3n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assay


J Med Chem 55: 6975-9 (2012)


Article DOI: 10.1021/jm300700v
BindingDB Entry DOI: 10.7270/Q2KD2017
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84167
PNG
(MLS000579971 | N-cyclohexyl-2-(4-fluoranylphenoxy)...)
Show SMILES Fc1ccc(OCC(=O)N(C2CCCCC2)c2ccccn2)cc1
Show InChI InChI=1S/C19H21FN2O2/c20-15-9-11-17(12-10-15)24-14-19(23)22(16-6-2-1-3-7-16)18-8-4-5-13-21-18/h4-5,8-13,16H,1-3,6-7,14H2
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n/an/a 1.49E+3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM84192
PNG
(MLS001160615 | SMR000709152 | [2-(3,4-dimethoxyphe...)
Show SMILES COc1ccc(cc1OC)-c1cc(C(=O)N2CC(C)CC(C)C2)c2ccccc2n1
Show InChI InChI=1S/C25H28N2O3/c1-16-11-17(2)15-27(14-16)25(28)20-13-22(26-21-8-6-5-7-19(20)21)18-9-10-23(29-3)24(12-18)30-4/h5-10,12-13,16-17H,11,14-15H2,1-4H3
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n/an/a 1.51E+3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv7.2


(Rattus norvegicus)
BDBM77218
PNG
(2-[(5-methyl-2-p-phenetyl-oxazol-4-yl)methylthio]-...)
Show SMILES CCOc1ccc(cc1)-c1nc(CSCC(=O)NC2CCCc3ccccc23)c(C)o1
Show InChI InChI=1S/C25H28N2O3S/c1-3-29-20-13-11-19(12-14-20)25-27-23(17(2)30-25)15-31-16-24(28)26-22-10-6-8-18-7-4-5-9-21(18)22/h4-5,7,9,11-14,22H,3,6,8,10,15-16H2,1-2H3,(H,26,28)
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n/an/a 1.51E+3n/an/an/an/an/an/a



Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay


Assay Description
Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC_KCNQ2_Inh_HFCP_IWS_CRC) Center Affiliation: Johns Hopkins University, School of M...


PubChem Bioassay (2011)


BindingDB Entry DOI: 10.7270/Q2W37TT2
More data for this
Ligand-Target Pair
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