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Found 14 Enz. Inhib. hit(s) with all data for entry = 813
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292143(2-(2-((2,3-dihydrobenzo[b][1,4]dioxo-6-yl)oxy)-5-h...)
Affinity DataIC50:  210nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292144(2-(2-([1,1′-biphenyl]-4-oxo)-5-hydroxy-8-met...)
Affinity DataIC50:  230nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292141((2-(2-(4-bromophenoxy)-5-hydroxy-8-methyl-1,7-naph...)
Affinity DataIC50:  330nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292142(2-(2-(3-(tert-butyl)phenoxy)-5-hydroxy-8-methyl-1,...)
Affinity DataIC50:  510nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292145(2-(5-hydroxy-2-(4-methoxyphenoxy)-8-methyl-1,7-nap...)
Affinity DataIC50:  1.40E+3nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292135(2-(2-(4-cyanophenoxy)-5-hydroxy-8-methyl-1,7-napht...)
Affinity DataIC50:  2.20E+3nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292138(2-(2-(4-chlorophenoxy)-5-hydroxy-8-methyl-1,7-naph...)
Affinity DataIC50:  4.00E+3nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292140(2-(2-(3-cyanophenoxy)-5-hydroxy-8-methyl-1,7-napht...)
Affinity DataIC50:  5.10E+3nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292137(2-(5-hydroxy-2-phenoxy-1,7-naphthyridine-6-formami...)
Affinity DataIC50:  6.90E+3nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292132(2-(5-hydroxy-8-methyl-2-phenoxy-1,7-naphthyridine-...)
Affinity DataIC50:  3.30E+4nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292139((2-5-hydroxy-8-methyl-2-(4-(trifluoromethyl)phenox...)
Affinity DataIC50:  3.60E+4nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292134(2-(2-(3-chlorophenoxy)-5-hydroxy-8-methyl-1,7-naph...)
Affinity DataIC50:  4.80E+4nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292136(2-(2-(4-(tert-butyl)phenoxy)-5-hydroxy-8-methyl-1,...)
Affinity DataIC50:  5.90E+4nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1(Homo sapiens (Human))
Shenyang Sunshine Pharmaceutical

US Patent
LigandPNGBDBM292133((2-(2-(4-fluorophenoxy)-5-hydroxy-8-methyl-1,7-nap...)
Affinity DataIC50:  7.30E+4nMT: 2°CAssay Description:To a NETN (20 mM Tris.HCl, 100 mM NaCl, 1 mM EDTA, 0.5% NP-40, 1 mM PMSF) buffer containing 200 μM ascorbic acid, 20 μM α-ketoglutaric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent