Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 884
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296828(1-(2-(Difluoromethoxy)phenyl)-8-(6-methoxypyridin-...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296866(1-(2-(Difluoromethoxy)phenyl)-4-methyl-8-(1-methyl...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296838(1-(2,5-Dimethylphenyl)-8-(1-methyl-1H-pyrazol-4-yl...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296864(1-(2-(Difluoromethoxy)phenyl)-8-(6-methoxypyridin-...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296863(1-(2,5-Dimethylphenyl)-8-(6-methoxypyridin-3-yl)-4...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296861(2-(4-(1-(2-(Difluoromethoxy)phenyl)-1,2,3,4-tetrah...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296860(2-(5-(1-(2-(Difluoromethoxy)phenyl)-1,2,3,4-tetrah...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296840(4-(5-(1-(2,5-Dimethylphenyl)-1,2,3,4-tetrahydroimi...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296858(1-(5-Chloro-2-methylphenyl)-8-(6-methoxypyridin-3-...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296857(1-(2-Chlorophenyl)-8-(6-methoxypyridin-3-yl)-1,2,3...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296829(1-(2,5-Dimethylphenyl)-7-methyl-8-(1-methyl-1H-pyr...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296831(1-(2,5-Dimethylphenyl)-8-(6-methoxypyridin-3-yl)-1...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296832(1-(2-(Difluoromethoxy)phenyl)-8-(6-methoxypyridin-...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296833(1-(2-Methoxy-5-methylphenyl)-8-(6-methoxypyridin-3...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296835(8-(6-Methoxypyridin-3-yl)-1-(o-tolyl)-1,2,3,4-tetr...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296836(8-(6-Methoxypyridin-3-yl)-1-(2-(trifluoromethoxy)p...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296838(1-(2,5-Dimethylphenyl)-8-(1-methyl-1H-pyrazol-4-yl...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296839(1-(2-(Difluoromethoxy)phenyl)-8-(1-methyl-1H-pyraz...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296840(4-(5-(1-(2,5-Dimethylphenyl)-1,2,3,4-tetrahydroimi...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296841(4-(5-(1-(2-(Difluoromethoxy)phenyl)-1,2,3,4-tetrah...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296842(2-(4-(1-(2,5-Dimethylphenyl)-1,2,3,4-tetrahydroimi...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296843(2-(4-(1-(2-(Difluoromethoxy)phenyl)-1,2,3,4-tetrah...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296844(2-(5-(1-(2,5-Dimethylphenyl)-1,2,3,4-tetrahydroimi...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296845(4-(5-(1-(2-(Difluoromethoxy)-5-methylphenyl)-1,2,3...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296846(1-(2-(Difluoromethoxy)-5-methylphenyl)-8-(6-methox...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296847(2-(5-(7-Chloro-1-phenyl-1,2,3,4-tetrahydroimidazo[...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296851(1-(5-Fluoro-2-methylphenyl)-8-(6-methoxypyridin-3-...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296852(1-(4-Fluoro-2-methylphenyl)-8-(6-methoxypyridin-3-...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296833(1-(2-Methoxy-5-methylphenyl)-8-(6-methoxypyridin-3...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296854(1-(2-Ethylphenyl)-8-(6-methoxypyridin-3-yl)-1,2,3,...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296836(8-(6-Methoxypyridin-3-yl)-1-(2-(trifluoromethoxy)p...)
Affinity DataIC50: <1.00E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296856(1-(2,4-Dimethylphenyl)-8-(6-methoxypyridin-3-yl)-1...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296862(2-(4-(1-(2,5-Dimethylphenyl)-1,2,3,4-tetrahydroimi...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296834(1-(Isoquinolin-1-yl)-8-(6-methoxypyridin-3-yl)-1,2...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296850(1-(2,3-Dimethylphenyl)-8-(6-methoxypyridin-3-yl)-1...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296827(1-(2,5-Dimethylphenyl)-8-(6-methoxypyridin-3-yl)-7...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296848(7-Chloro-1-(2-(difluoromethoxy)phenyl)-8-(6-methox...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296830(1-(2-(Difluoromethoxy)phenyl)-7-methyl-8-(1-methyl...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296837(8-(6-Methoxypyridin-3-yl)-1-(2-methyl-5-(trifluoro...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296867(4-(5-(1-(2,5-Dimethylphenyl)-6,7-dimethyl-1,2,3,4-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM296849(7-Chloro-1-(2,5-dimethylphenyl)-8-(6-methoxypyridi...)
Affinity DataIC50:  5.50E+3nMAssay Description:Test compounds serially diluted in DMSO were plated in an assay plate (Labcyte, Cat. #LP-0200) at final concentrations ranging from 0.004 μM to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent