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Found 17 Enz. Inhib. hit(s) with all data for entry = 1375
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318948(2-Methyl-2-[[7-(4-nitrophenyl)benzo[d]isothiazol-6...)
Affinity DataIC50:  12nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318954(2-[[7-(4-Cyanophenyl)benzo[d]isothiazol-6-yl]thio]...)
Affinity DataIC50:  21nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318946(1-[[7-(4-Cyanophenyl)benzo[d]isothiazol-6-yl]thio]...)
Affinity DataIC50:  21.5nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318956((E)-3-[[1-(4-cyanophenyl)naphthalen-2-yl]thio]-2-b...)
Affinity DataIC50:  25nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318947(1-[[7-(4-Cyanophenyl)benzo[d]isothiazol-6-yl]thio]...)
Affinity DataIC50:  26.2nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318949(2-Methyl-2-[[7-[4-(trifluoromethyl)phenyl]benzo[d]...)
Affinity DataIC50:  104nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318950(2-[[7-(4-Chlorophenyl)benzo[d]isothiazol-6-yl]thio...)
Affinity DataIC50:  106nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318952(2-[[7-(4-Cyano-3-fluorophenyl)benzo[d]isothiazol-6...)
Affinity DataIC50:  161nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318944(2-[[7-(4-Cyanophenyl)benzo[d]thiazol-6-yl]thio]-2-...)
Affinity DataIC50:  170nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318951(2-[[7-(3-Cyanophenyl)benzo[d]isothiazol-6-yl]thio]...)
Affinity DataIC50:  205nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318957(1-[[7-(4-Cyanophenyl)benzo[d]isothazol-6-yl]thio]c...)
Affinity DataIC50:  296nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318955(2-[[7-(4-Cyanophenyl)benzo[d]isothiazol-6-yl]thio]...)
Affinity DataIC50:  474nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318942(2-[(4′-Cyano[1,1′-binaphthalene]-2-yl)...)
Affinity DataIC50:  790nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318945(2-[[3-(4-Cyanophenyl)quinolin-4-yl]thio]-2-methylp...)
Affinity DataIC50:  1.58E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318941(2-[(4′-Cyano-(1,1′-binaphthalene)-2-yl...)
Affinity DataIC50:  2.06E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318953(1-[[7-(4-Cyanophenyl)-3-methylbenzo[d]isothiazol-6...)
Affinity DataIC50:  2.43E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Nippon Chemiphar

US Patent
LigandPNGBDBM318943(2-[[5-(4-Cyanophenyl)quinolin-6-yl]thio]-2-methylp...)
Affinity DataIC50:  3.44E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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