Compile Data Set for Download or QSAR
maximum 50k data
Found 605 Enz. Inhib. hit(s) with all data for entry = 5611
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405060(1-[2-fluoro-4-(4-{2-[2-fluoro-5- (trifluoromethoxy...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405061(1-(2-fluoro-4-{4-[2-(6-methylpyridin- 3-yl)acetami...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405062(1-[2-fluoro-4-(4-{2-[3- (trifluoromethoxy)phenyl]a...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405063(1-[2-fluoro-4-(4-{2-[3- (trifluoromethoxy)phenyl]a...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405064(1-[2-fluoro-4-(4-{2-[3- (trifluoromethoxy)phenyl]a...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405067(1-[3-fluoro-4-(4-{2-[3- (trifluoromethoxy)phenyl]a...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405068(1-[3-fluoro-4-(4-{2-[2-fluoro-5- (trifluoromethoxy...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405069(1-[4-(4-{2-[2-fluoro-5- (trifluoromethoxy)phenyl]a...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405070(1-[4-(4-{2-[3- (trifluoromethoxy)phenyl]acetamido}...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405071(1-(4-{4-[2-(5-chloro-2- fluorophenyl)acetamido]-1H...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405072(1-[2-fluoro-4-(4-{2-[2-fluoro-5- (trifluoromethoxy...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405073(1-[2-fluoro-4-(4-{2-[2-fluoro-5- (trifluoromethoxy...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405069(1-[4-(4-{2-[2-fluoro-5- (trifluoromethoxy)phenyl]a...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405075(1-(2-fluoro-4-{4-[2-(pyridin-2- yl)acetamido]-1H-1...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405076(5-[3-fluoro-4-(4-{[(6-methylpyridin- 3-yl)methyl]c...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405077(1-{2-fluoro-4-[4-({[6- (trifluoromethyl)pyridin-3-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405078(1-{2-fluoro-4-[4-({[6- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405079(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405080(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405081(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405082(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405083(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405084(1-{2-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405085(1-{2-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405086(1-{2-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405087(1-{2-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405088(1-{2-fluoro-4-[4-({[4- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405089(1-{2-fluoro-4-[4-({[5- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405090(1-[2-fluoro-4-(4-{[(6-methylpyridin- 3-yl)methyl]c...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405091(1-{2-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405092(1-{2-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405093(1-{3-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405094(1-{3-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405095(1-{3-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405096(1-{3-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405097(1-{2-fluoro-4-[4-({[5- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405098(5-{3-fluoro-4-[4-({[3- (trifluoromethoxy)phenyl]me...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405099(5-{3-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405100(1-{3-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405101(5-{3-fluoro-4-[4-({[5- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405102(5-{3-fluoro-4-[4-({[4- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405103(5-[3-fluoro-4-(4-{[(6-methylpyridin- 3-yl)methyl]c...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405104(5-{3-fluoro-4-[4-({[5- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405105(5-{3-fluoro-4-[4-({[4- (trifluoromethyl)pyridin-2-...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405106(N-benzyl-1-{2-fluoro-4-[4-({[4- (trifluoromethyl)p...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405107(5-{3-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405108(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405109(1-{2-fluoro-4-[4-({[2-fluoro-5- (trifluoromethoxy)...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405110(1-[2-fluoro-4-(4-{[(2- fluorophenyl)methyl]carbamo...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM405111(1-{2-fluoro-4-[4-({[3- (trifluoromethyl)phenyl]met...)
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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