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Found 85 Enz. Inhib. hit(s) with all data for entry = 8729
LigandPNGBDBM414876(4-Chloro-2-fluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[...)
Affinity DataIC50:  98nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414839((3S,4S)—N-(4-chlorophenyl)-N,3-dimethyl-1-[(2R)-3,...)
Affinity DataIC50:  110nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414842((3S,4S)—N-(2-fluoro-4-methylphenyl)-N,3-dimethyl-1...)
Affinity DataIC50:  120nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414853(N,4-Dimethyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,3-tri...)
Affinity DataIC50:  130nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414870(2-Chloro-4-fluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[...)
Affinity DataIC50:  150nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414836((3S,4S)—N,3-Dimethyl-N-(4-methylphenyl)-1-[(2R)-3,...)
Affinity DataIC50:  160nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414862(2,4-Difluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-...)
Affinity DataIC50:  180nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414831(1-((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-propiony...)
Affinity DataIC50:  200nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414841(N-(2-fluoro-4-methylphenyl)-N,3-dimethyl-1-[(2R)-3...)
Affinity DataIC50:  200nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414874(N,1-Dimethyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,3-tri...)
Affinity DataIC50:  230nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414868(2-Fluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  230nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414835(N,3-Dimethyl-N-(4-methylphenyl)-1-[(2R)-3,3,3-trif...)
Affinity DataIC50:  240nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414864(3,5-Difluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-...)
Affinity DataIC50:  240nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414856(4-Fluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  250nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414847(N,4-Dimethyl-N-{1-[(2R)-3,3,3-trifluoro-2-hydroxy-...)
Affinity DataIC50:  250nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414851(4-Chloro-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  260nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414848(2-Fluoro-4,N-dimethyl-N-{1-[(R)-3,3,3-trifluoro-2-...)
Affinity DataIC50:  260nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414838(N-(4-chlorophenyl)-N,3-dimethyl-1-[(2R)-3,3,3-trif...)
Affinity DataIC50:  270nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414878(N-Methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,3-trifluo...)
Affinity DataIC50:  290nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414866(4-Cyano-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,3...)
Affinity DataIC50:  300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414855(2-Fluoro-N,4-dimethyl-N-[(3R,4S)-3-methyl-1-[(2R)-...)
Affinity DataIC50:  300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414860(4-Methoxy-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3...)
Affinity DataIC50:  310nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414846(4-Chloro-N-methyl-N-{1-[(2R)-3,3,3-trifluoro-2-hyd...)
Affinity DataIC50:  390nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414880(N-Ethyl-2-fluoro-4-methyl-N-[1-((R)-3,3,3-trifluor...)
Affinity DataIC50:  410nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414832(1-((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-propiony...)
Affinity DataIC50:  410nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414872(5-Fluoro-N-methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  410nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414849(2-Chloro-N-methyl-N-{1-[(2R)-3,3,3-trifluoro-2-hyd...)
Affinity DataIC50:  550nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414834(1-((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-propiony...)
Affinity DataIC50:  590nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414858(N-Methyl-N-[(3R,4S)-3-methyl-1-[(2R)-3,3,3-trifluo...)
Affinity DataIC50:  710nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414843((3R,4R)—N-(2-fluoro-4-methylphenyl)-N,3-dimethyl-1...)
Affinity DataIC50:  770nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414830(1-((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-propiony...)
Affinity DataIC50:  1.10E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414861(4-Methoxy-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3...)
Affinity DataIC50:  1.30E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414881(2-Fluoro-N-isopropyl-4-methyl-N-[1-((R)-3,3,3-trif...)
Affinity DataIC50:  1.30E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414833(1-((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-propiony...)
Affinity DataIC50:  1.50E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414883(4-Cyano-N-isopropyl-N-[1-((R)-3,3,3-trifluoro-2-hy...)
Affinity DataIC50:  1.60E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414844(N-[2-chloro-4-(trifluoromethyl)phenyl]-N,3-dimethy...)
Affinity DataIC50:  1.70E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414882(4-Cyano-N-ethyl-N-[1-((R)-3,3,3-trifluoro-2-hydrox...)
Affinity DataIC50:  2.10E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414869(2-Fluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  2.40E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414865(3,5-Difluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-...)
Affinity DataIC50:  2.40E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414854(N,4-Dimethyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,3-tri...)
Affinity DataIC50:  2.70E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414879(N-Methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,3-trifluo...)
Affinity DataIC50:  2.90E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414859(N-Methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,3-trifluo...)
Affinity DataIC50:  3.40E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414871(2-Chloro-4-fluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[...)
Affinity DataIC50:  3.60E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414840((3R,4R)—N-(4-chlorophenyl)-N,3-dimethyl-1-[(2R)-3,...)
Affinity DataIC50:  3.80E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414877(4-Chloro-2-fluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[...)
Affinity DataIC50:  3.90E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414863(2,4-Difluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-...)
Affinity DataIC50:  4.90E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414837((3R,4R)—N,3-Dimethyl-N-(4-methylphenyl)-1-[(2R)-3,...)
Affinity DataIC50:  5.10E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414852(4-Chloro-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  5.90E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM414857(4-Fluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  7.90E+3nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM414873(5-Fluoro-N-methyl-N-[(3S,4R)-3-methyl-1-[(2R)-3,3,...)
Affinity DataIC50:  1.30E+4nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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